Affinity Data by PubMed id=22137786

PubMed code 22137786

Found 9 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Amine oxidase [flavin-containing] B (Homo sapiens (Human))	BDBM15579 (CHEMBL972 \| DEPRENYL \| L-Deprenyl \| N-methyl-N-[(2...) Show SMILES C[C@H](Cc1ccccc1)N(C)CC#C \|r\| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	17	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ degli Studi di Cagliari Curated by ChEMBL					Assay Description Inhibition of human recombinant MAOB expressed in baculovirus-infected BTI insect cells assessed as using transformed p-tyramine after 15 mins by flu...				Bioorg Med Chem Lett 22: 258-61 (2011) Article DOI: 10.1016/j.bmcl.2011.11.020 BindingDB Entry DOI: 10.7270/Q2TH8N4X
Universit£ degli Studi di Cagliari Curated by ChEMBL					More data for this Ligand-Target Pair
Amine oxidase [flavin-containing] B (Homo sapiens (Human))	BDBM50360811 (CHEMBL1934677) Show SMILES COc1ccc(cc1Cl)-c1c(O)c2cc(Cl)ccc2oc1=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.79E+3	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ degli Studi di Cagliari Curated by ChEMBL					Assay Description Inhibition of human recombinant MAOB expressed in baculovirus-infected BTI insect cells assessed as using transformed p-tyramine after 15 mins by flu...				Bioorg Med Chem Lett 22: 258-61 (2011) Article DOI: 10.1016/j.bmcl.2011.11.020 BindingDB Entry DOI: 10.7270/Q2TH8N4X
Universit£ degli Studi di Cagliari Curated by ChEMBL					More data for this Ligand-Target Pair
Amine oxidase [flavin-containing] A (Homo sapiens (Human))	BDBM29136 (CHEMBL92401 \| Euphozid \| Iprazid \| Iproniazid) Show SMILES CC(C)NNC(=O)c1ccncc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	6.56E+3	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ degli Studi di Cagliari Curated by ChEMBL					Assay Description Inhibition of human recombinant MAOA expressed in baculovirus-infected BTI insect cells assessed as conversion of p-tyramine into p-hydroxyphenyl-ace...				Bioorg Med Chem Lett 22: 258-61 (2011) Article DOI: 10.1016/j.bmcl.2011.11.020 BindingDB Entry DOI: 10.7270/Q2TH8N4X
Universit£ degli Studi di Cagliari Curated by ChEMBL					More data for this Ligand-Target Pair
Amine oxidase [flavin-containing] B (Homo sapiens (Human))	BDBM29136 (CHEMBL92401 \| Euphozid \| Iprazid \| Iproniazid) Show SMILES CC(C)NNC(=O)c1ccncc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	7.54E+3	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ degli Studi di Cagliari Curated by ChEMBL					Assay Description Inhibition of human recombinant MAOB expressed in baculovirus-infected BTI insect cells assessed as using transformed p-tyramine after 15 mins by flu...				Bioorg Med Chem Lett 22: 258-61 (2011) Article DOI: 10.1016/j.bmcl.2011.11.020 BindingDB Entry DOI: 10.7270/Q2TH8N4X
Universit£ degli Studi di Cagliari Curated by ChEMBL					More data for this Ligand-Target Pair
Amine oxidase [flavin-containing] B (Homo sapiens (Human))	BDBM50360809 (CHEMBL1934675) Show SMILES COc1ccc(cc1Cl)-c1c(O)c2ccccc2oc1=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	9.26E+3	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ degli Studi di Cagliari Curated by ChEMBL					Assay Description Inhibition of human recombinant MAOB expressed in baculovirus-infected BTI insect cells assessed as using transformed p-tyramine after 15 mins by flu...				Bioorg Med Chem Lett 22: 258-61 (2011) Article DOI: 10.1016/j.bmcl.2011.11.020 BindingDB Entry DOI: 10.7270/Q2TH8N4X
Universit£ degli Studi di Cagliari Curated by ChEMBL					More data for this Ligand-Target Pair
Amine oxidase [flavin-containing] B (Homo sapiens (Human))	BDBM50360808 (CHEMBL1934673) Show SMILES COc1ccc(cc1)-c1c(O)c2cc(C)ccc2oc1=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.20E+4	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ degli Studi di Cagliari Curated by ChEMBL					Assay Description Inhibition of human recombinant MAOB expressed in baculovirus-infected BTI insect cells assessed as using transformed p-tyramine after 15 mins by flu...				Bioorg Med Chem Lett 22: 258-61 (2011) Article DOI: 10.1016/j.bmcl.2011.11.020 BindingDB Entry DOI: 10.7270/Q2TH8N4X
Universit£ degli Studi di Cagliari Curated by ChEMBL					More data for this Ligand-Target Pair
Amine oxidase [flavin-containing] B (Homo sapiens (Human))	BDBM50360810 (CHEMBL1934676) Show SMILES COc1ccc(cc1Cl)-c1c(O)c2cc(C)ccc2oc1=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.27E+4	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ degli Studi di Cagliari Curated by ChEMBL					Assay Description Inhibition of human recombinant MAOB expressed in baculovirus-infected BTI insect cells assessed as using transformed p-tyramine after 15 mins by flu...				Bioorg Med Chem Lett 22: 258-61 (2011) Article DOI: 10.1016/j.bmcl.2011.11.020 BindingDB Entry DOI: 10.7270/Q2TH8N4X
Universit£ degli Studi di Cagliari Curated by ChEMBL					More data for this Ligand-Target Pair
Amine oxidase [flavin-containing] A (Homo sapiens (Human))	BDBM15579 (CHEMBL972 \| DEPRENYL \| L-Deprenyl \| N-methyl-N-[(2...) Show SMILES C[C@H](Cc1ccccc1)N(C)CC#C \|r\| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	6.87E+4	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ degli Studi di Cagliari Curated by ChEMBL					Assay Description Inhibition of human recombinant MAOA expressed in baculovirus-infected BTI insect cells assessed as conversion of p-tyramine into p-hydroxyphenyl-ace...				Bioorg Med Chem Lett 22: 258-61 (2011) Article DOI: 10.1016/j.bmcl.2011.11.020 BindingDB Entry DOI: 10.7270/Q2TH8N4X
Universit£ degli Studi di Cagliari Curated by ChEMBL					More data for this Ligand-Target Pair
Amine oxidase [flavin-containing] B (Homo sapiens (Human))	BDBM50360807 (CHEMBL1917495) Show SMILES COc1ccc(cc1)-c1c(O)c2ccccc2oc1=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	6.96E+4	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ degli Studi di Cagliari Curated by ChEMBL					Assay Description Inhibition of human recombinant MAOB expressed in baculovirus-infected BTI insect cells assessed as using transformed p-tyramine after 15 mins by flu...				Bioorg Med Chem Lett 22: 258-61 (2011) Article DOI: 10.1016/j.bmcl.2011.11.020 BindingDB Entry DOI: 10.7270/Q2TH8N4X
Universit£ degli Studi di Cagliari Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%