Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50340226 (4-amino-1-((6-methylpyridin-3-yl)methyl)-6-(oxazol...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 100 | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Agonist activity at TLR7 | Bioorg Med Chem Lett 22: 2856-60 (2012) Article DOI: 10.1016/j.bmcl.2012.02.069 BindingDB Entry DOI: 10.7270/Q2KH0PC8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 7 (Homo sapiens (Human)) | BDBM50340220 (4-amino-1-((6-methylpyridin-3-yl)methyl)-6-(triflu...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 50 | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Agonist activity at TLR7 | Bioorg Med Chem Lett 22: 2856-60 (2012) Article DOI: 10.1016/j.bmcl.2012.02.069 BindingDB Entry DOI: 10.7270/Q2KH0PC8 | |||||||||||
More data for this Ligand-Target Pair |