Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Androgen receptor (Homo sapiens (Human)) | BDBM50398195 (CHEMBL2177238) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | 9.60 | n/a | n/a | n/a | n/a | n/a | n/a |
GALAPAGOS, Parc Biocitech Curated by ChEMBL | Assay Description Binding affinity to androgen receptor by competitive binding assay | J Med Chem 55: 8225-35 (2012) Article DOI: 10.1021/jm300249m BindingDB Entry DOI: 10.7270/Q2XW4KXM | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50398195 (CHEMBL2177238) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 8.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
GALAPAGOS, Parc Biocitech Curated by ChEMBL | Assay Description Binding affinity to progesterone receptor by competitive binding assay | J Med Chem 55: 8225-35 (2012) Article DOI: 10.1021/jm300249m BindingDB Entry DOI: 10.7270/Q2XW4KXM | |||||||||||
More data for this Ligand-Target Pair |