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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Melanin-concentrating hormone receptor 1 (RAT) | BDBM50391543 (CHEMBL2147477) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet  | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.10 | n/a | n/a | n/a | n/a | n/a | n/a |
LEO Pharma Curated by ChEMBL | Assay Description Antagonist activity at rat MCH1 receptor expressed in HEK 293T cells assessed as inhibition of MCH-induced Ca2+ mobilization after 10 mins by FLIPR a... | Bioorg Med Chem Lett 22: 6039-47 (2012) Article DOI: 10.1016/j.bmcl.2012.08.025 BindingDB Entry DOI: 10.7270/Q2T72JHK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Melanin-concentrating hormone receptor 1 (Homo sapiens (Human)) | BDBM50391542 (CHEMBL2147476) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
LEO Pharma Curated by ChEMBL | Assay Description Displacement of [125I]-MCH from human MCHR1 receptor expressed in CHO-K1 cell membranes after 2 hrs by scintillation proximity assay | Bioorg Med Chem Lett 22: 6039-47 (2012) Article DOI: 10.1016/j.bmcl.2012.08.025 BindingDB Entry DOI: 10.7270/Q2T72JHK | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
