Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50427063 (CHEMBL2322841) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.5 | n/a | n/a | n/a | n/a |
College of Pharmacy of Kangwon National University Curated by ChEMBL | Assay Description Agonist activity at human GPR119 transfected in HEK293 cells assessed as concentration for 50 % cAMP stimulation of oleylethanolamine | Bioorg Med Chem Lett 23: 1519-21 (2013) Article DOI: 10.1016/j.bmcl.2012.12.011 BindingDB Entry DOI: 10.7270/Q2SQ91Q7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50427061 (CHEMBL2322839) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 6.70 | n/a | n/a | n/a | n/a |
College of Pharmacy of Kangwon National University Curated by ChEMBL | Assay Description Agonist activity at human GPR119 transfected in HEK293 cells assessed as concentration for 50 % cAMP stimulation of oleylethanolamine | Bioorg Med Chem Lett 23: 1519-21 (2013) Article DOI: 10.1016/j.bmcl.2012.12.011 BindingDB Entry DOI: 10.7270/Q2SQ91Q7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50427059 (CHEMBL2322837) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.5 | n/a | n/a | n/a | n/a |
College of Pharmacy of Kangwon National University Curated by ChEMBL | Assay Description Agonist activity at human GPR119 transfected in HEK293 cells assessed as concentration for 50 % cAMP stimulation of oleylethanolamine | Bioorg Med Chem Lett 23: 1519-21 (2013) Article DOI: 10.1016/j.bmcl.2012.12.011 BindingDB Entry DOI: 10.7270/Q2SQ91Q7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50427060 (CHEMBL2322838) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.90 | n/a | n/a | n/a | n/a |
College of Pharmacy of Kangwon National University Curated by ChEMBL | Assay Description Agonist activity at human GPR119 transfected in HEK293 cells assessed as concentration for 50 % cAMP stimulation of oleylethanolamine | Bioorg Med Chem Lett 23: 1519-21 (2013) Article DOI: 10.1016/j.bmcl.2012.12.011 BindingDB Entry DOI: 10.7270/Q2SQ91Q7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50427062 (CHEMBL2322840) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
College of Pharmacy of Kangwon National University Curated by ChEMBL | Assay Description Agonist activity at human GPR119 transfected in HEK293 cells assessed as concentration for 50 % cAMP stimulation of oleylethanolamine | Bioorg Med Chem Lett 23: 1519-21 (2013) Article DOI: 10.1016/j.bmcl.2012.12.011 BindingDB Entry DOI: 10.7270/Q2SQ91Q7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM29080 (CHEMBL280065 | N-oleoylethanolamine | Oleamide MEA...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.20E+3 | n/a | n/a | n/a | n/a |
College of Pharmacy of Kangwon National University Curated by ChEMBL | Assay Description Agonist activity at human GPR119 transfected in HEK293 cells assessed as concentration for 50 % cAMP stimulation of oleylethanolamine | Bioorg Med Chem Lett 23: 1519-21 (2013) Article DOI: 10.1016/j.bmcl.2012.12.011 BindingDB Entry DOI: 10.7270/Q2SQ91Q7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50427060 (CHEMBL2322838) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 15 | n/a | n/a | n/a | n/a |
College of Pharmacy of Kangwon National University Curated by ChEMBL | Assay Description Agonist activity at human GPR119 transfected in HEK293 cells assessed as concentration for 50 % cAMP stimulation of oleylethanolamine | Bioorg Med Chem Lett 23: 1519-21 (2013) Article DOI: 10.1016/j.bmcl.2012.12.011 BindingDB Entry DOI: 10.7270/Q2SQ91Q7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50427059 (CHEMBL2322837) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a |
College of Pharmacy of Kangwon National University Curated by ChEMBL | Assay Description Agonist activity at human GPR119 transfected in HEK293 cells assessed as concentration for 50 % cAMP stimulation of oleylethanolamine | Bioorg Med Chem Lett 23: 1519-21 (2013) Article DOI: 10.1016/j.bmcl.2012.12.011 BindingDB Entry DOI: 10.7270/Q2SQ91Q7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50427064 (CHEMBL2322842) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 12 | n/a | n/a | n/a | n/a |
College of Pharmacy of Kangwon National University Curated by ChEMBL | Assay Description Agonist activity at human GPR119 transfected in HEK293 cells assessed as concentration for 50 % cAMP stimulation of oleylethanolamine | Bioorg Med Chem Lett 23: 1519-21 (2013) Article DOI: 10.1016/j.bmcl.2012.12.011 BindingDB Entry DOI: 10.7270/Q2SQ91Q7 | |||||||||||
More data for this Ligand-Target Pair |