Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glutamate receptor 2 (Homo sapiens (Human)) | BDBM50427677 (CHEMBL2323527) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 5.60E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Yokohama City University Curated by ChEMBL | Assay Description Binding affinity to GluA2 ligand binding domain (unknown origin) by competitive binding assay | J Med Chem 56: 2283-93 (2013) Article DOI: 10.1021/jm301590z BindingDB Entry DOI: 10.7270/Q2SJ1MZN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 2 (Rattus norvegicus) | BDBM50178141 ((S)-1-(2-amino-2-carboxyethyl)-3-(4-carboxybenzyl)...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Similars | MMDB PDB Article PubMed | n/a | n/a | 2.90E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Yokohama City University Curated by ChEMBL | Assay Description Displacement of [3H]AMPA from rat GluA2 ligand binding domain after 1 hr | J Med Chem 56: 2283-93 (2013) Article DOI: 10.1021/jm301590z BindingDB Entry DOI: 10.7270/Q2SJ1MZN | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |