Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50094064 (CHEMBL335799 | GSS(heptyl carbonyl)F-NH2) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 72 | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Milano Curated by ChEMBL | Assay Description Agonist activity at GHS-R1a (unknown origin) | Bioorg Med Chem 21: 5470-9 (2013) Article DOI: 10.1016/j.bmc.2013.06.006 BindingDB Entry DOI: 10.7270/Q2VQ3446 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50438564 (CHEMBL2413152) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.600 | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Milano Curated by ChEMBL | Assay Description Agonist activity at GHS-R1a (unknown origin) | Bioorg Med Chem 21: 5470-9 (2013) Article DOI: 10.1016/j.bmc.2013.06.006 BindingDB Entry DOI: 10.7270/Q2VQ3446 | |||||||||||
More data for this Ligand-Target Pair |