Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50442743 (CHEMBL2442998) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Bari 'Aldo Moro' Curated by ChEMBL | Assay Description Binding affinity to sigma 1 receptor (unknown origin) by radioligand binding assay | Bioorg Med Chem Lett 23: 6083-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.025 BindingDB Entry DOI: 10.7270/Q23T9JPT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50442745 (CHEMBL2442996) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Bari 'Aldo Moro' Curated by ChEMBL | Assay Description Binding affinity to sigma 1 receptor (unknown origin) by radioligand binding assay | Bioorg Med Chem Lett 23: 6083-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.025 BindingDB Entry DOI: 10.7270/Q23T9JPT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50442742 (CHEMBL2442999) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Bari 'Aldo Moro' Curated by ChEMBL | Assay Description Binding affinity to sigma 1 receptor (unknown origin) by radioligand binding assay | Bioorg Med Chem Lett 23: 6083-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.025 BindingDB Entry DOI: 10.7270/Q23T9JPT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50442744 (CHEMBL2442997) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Bari 'Aldo Moro' Curated by ChEMBL | Assay Description Binding affinity to sigma 1 receptor (unknown origin) by radioligand binding assay | Bioorg Med Chem Lett 23: 6083-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.025 BindingDB Entry DOI: 10.7270/Q23T9JPT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50253281 (CHEMBL522691 | N-(4-Cyanophenylmethyl)-4-(2-diphen...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Bari 'Aldo Moro' Curated by ChEMBL | Assay Description Binding affinity to sigma 1 receptor (unknown origin) by radioligand binding assay | Bioorg Med Chem Lett 23: 6083-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.025 BindingDB Entry DOI: 10.7270/Q23T9JPT | |||||||||||
More data for this Ligand-Target Pair |