Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
BDNF/NT-3 growth factors receptor (Homo sapiens (Human)) | BDBM50093539 (7,8-Dihydroxy-2-phenyl-chromen-4-one | 7,8-Dihydro...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | 320 | n/a | n/a | n/a | n/a | n/a |
Universit£ de Montr£al Curated by ChEMBL | Assay Description Binding affinity to TrkB receptor extracellular domain (unknown origin) after 10 mins by liquid Scatchard plot analysis | Bioorg Med Chem 21: 7816-29 (2013) Article DOI: 10.1016/j.bmc.2013.10.012 BindingDB Entry DOI: 10.7270/Q2BV7J3Z | |||||||||||
More data for this Ligand-Target Pair |