Affinity Data by PubMed id=24368028

PubMed code 24368028

Found 4 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Glutamate receptor ionotropic, kainate 2 (Homo sapiens (Human))	BDBM50445689 (CHEMBL3104225) Show SMILES CCn1c(c(C)c2cc(OC)ccc12)-c1ccc(OC)cc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	700	n/a	n/a	n/a	n/a	n/a	n/a
Medical University of Lublin Curated by ChEMBL					Assay Description Displacement of [3H]-kainate from GluK2 receptor (unknown origin)				Bioorg Med Chem 22: 787-95 (2014) Article DOI: 10.1016/j.bmc.2013.12.013 BindingDB Entry DOI: 10.7270/Q2C82BS0
Medical University of Lublin Curated by ChEMBL					More data for this Ligand-Target Pair
Glutamate receptor ionotropic, kainate 2 (Homo sapiens (Human))	BDBM50445686 (CHEMBL3104264) Show SMILES CCn1c(c(C)c2cc(OC)ccc12)-c1ccccc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	6.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Medical University of Lublin Curated by ChEMBL					Assay Description Displacement of [3H]-kainate from GluK2 receptor (unknown origin)				Bioorg Med Chem 22: 787-95 (2014) Article DOI: 10.1016/j.bmc.2013.12.013 BindingDB Entry DOI: 10.7270/Q2C82BS0
Medical University of Lublin Curated by ChEMBL					More data for this Ligand-Target Pair
Glutamate receptor ionotropic, kainate 2 (Homo sapiens (Human))	BDBM50445688 (CHEMBL3104262) Show SMILES CCn1c(cc2cc(OC)ccc12)-c1ccccc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	6.70E+3	n/a	n/a	n/a	n/a	n/a	n/a
Medical University of Lublin Curated by ChEMBL					Assay Description Displacement of [3H]-kainate from GluK2 receptor (unknown origin)				Bioorg Med Chem 22: 787-95 (2014) Article DOI: 10.1016/j.bmc.2013.12.013 BindingDB Entry DOI: 10.7270/Q2C82BS0
Medical University of Lublin Curated by ChEMBL					More data for this Ligand-Target Pair
Glutamate receptor ionotropic, kainate 2 (Homo sapiens (Human))	BDBM50445687 (CHEMBL3104263) Show SMILES CCn1c(c(C)c2ccccc12)-c1ccc(OC)cc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Medical University of Lublin Curated by ChEMBL					Assay Description Displacement of [3H]-kainate from GluK2 receptor (unknown origin)				Bioorg Med Chem 22: 787-95 (2014) Article DOI: 10.1016/j.bmc.2013.12.013 BindingDB Entry DOI: 10.7270/Q2C82BS0
Medical University of Lublin Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%