Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Oxa40 (Acinetobacter baumannii) | BDBM227598 (Penem 1) | PDB MMDB KEGG UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 30 | n/a | 150 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Case Western Reserve University | Assay Description Steady-state kinetics were performed on an Agilent 8453 diode array spectrophotometer (Palo Alto, CA) in 50 mM sodium phosphate buffer (pH 7.2) suppl... | J Biol Chem 289: 6152-64 (2014) Article DOI: 10.1074/jbc.M113.533562 BindingDB Entry DOI: 10.7270/Q2CN72SC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-lactamase OXA-1 (Escherichia coli (Enterobacteria)) | BDBM227598 (Penem 1) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 50 | n/a | 30 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Case Western Reserve University | Assay Description Steady-state kinetics were performed on an Agilent 8453 diode array spectrophotometer (Palo Alto, CA) in 50 mM sodium phosphate buffer (pH 7.2) suppl... | J Biol Chem 289: 6152-64 (2014) Article DOI: 10.1074/jbc.M113.533562 BindingDB Entry DOI: 10.7270/Q2CN72SC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxa40 (Acinetobacter baumannii) | BDBM227599 (Penem 3) | PDB MMDB KEGG UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 150 | n/a | 160 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Case Western Reserve University | Assay Description Steady-state kinetics were performed on an Agilent 8453 diode array spectrophotometer (Palo Alto, CA) in 50 mM sodium phosphate buffer (pH 7.2) suppl... | J Biol Chem 289: 6152-64 (2014) Article DOI: 10.1074/jbc.M113.533562 BindingDB Entry DOI: 10.7270/Q2CN72SC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-lactamase OXA-1 (Escherichia coli (Enterobacteria)) | BDBM227599 (Penem 3) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 380 | n/a | 60 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Case Western Reserve University | Assay Description Steady-state kinetics were performed on an Agilent 8453 diode array spectrophotometer (Palo Alto, CA) in 50 mM sodium phosphate buffer (pH 7.2) suppl... | J Biol Chem 289: 6152-64 (2014) Article DOI: 10.1074/jbc.M113.533562 BindingDB Entry DOI: 10.7270/Q2CN72SC | |||||||||||
More data for this Ligand-Target Pair |