Affinity Data by PubMed id=24900220

PubMed code 24900220

Found 9 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Signal transducer and activator of transcription 3 (Homo sapiens (Human))	BDBM50338992 (CHEMBL1687978 \| N-[5-(2-Furyl)-1,3,4-oxadiazol-2-y...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	5.50E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Inhibition of STAT3 transcriptional activity in human HeLa cells by luciferase reporter gene assay				ACS Med Chem Lett 1: 371-375 (2010) Article DOI: 10.1021/ml1000273 BindingDB Entry DOI: 10.7270/Q2FJ2H21
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Signal transducer and activator of transcription 3 (Homo sapiens (Human))	BDBM50338996 (2-(4-Chlorophenyl)-N-(5-phenyl-1,3,4-oxadiazol-2-y...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	6.10E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Inhibition of STAT3 transcriptional activity in human HeLa cells by luciferase reporter gene assay				ACS Med Chem Lett 1: 371-375 (2010) Article DOI: 10.1021/ml1000273 BindingDB Entry DOI: 10.7270/Q2FJ2H21
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Signal transducer and activator of transcription 3 (Homo sapiens (Human))	BDBM50338994 (CHEMBL1687976 \| N-[5-(2-Furyl)-1,3,4-oxadiazol-2-y...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	6.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Inhibition of STAT3 transcriptional activity in human HeLa cells by luciferase reporter gene assay				ACS Med Chem Lett 1: 371-375 (2010) Article DOI: 10.1021/ml1000273 BindingDB Entry DOI: 10.7270/Q2FJ2H21
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Signal transducer and activator of transcription 3 (Homo sapiens (Human))	BDBM50338995 (2-Phenyl-N-(5-phenyl-1,3,4-oxadiazol-2-yl)-4-quino...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	6.60E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Inhibition of STAT3 transcriptional activity in human HeLa cells by luciferase reporter gene assay				ACS Med Chem Lett 1: 371-375 (2010) Article DOI: 10.1021/ml1000273 BindingDB Entry DOI: 10.7270/Q2FJ2H21
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Signal transducer and activator of transcription 3 (Homo sapiens (Human))	BDBM50338993 (2-(2-Furyl)-N-[5-(2-furyl)-1,3,4-oxadiazol-2-yl]-4...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	6.60E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Inhibition of STAT3 transcriptional activity in human HeLa cells by luciferase reporter gene assay				ACS Med Chem Lett 1: 371-375 (2010) Article DOI: 10.1021/ml1000273 BindingDB Entry DOI: 10.7270/Q2FJ2H21
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Signal transducer and activator of transcription 3 (Homo sapiens (Human))	BDBM50338998 (CHEMBL1687965 \| N-[5-(3-Furyl)-1,3,4-oxadiazol-2-y...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	7.20E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Inhibition of STAT3 transcriptional activity in human HeLa cells by luciferase reporter gene assay				ACS Med Chem Lett 1: 371-375 (2010) Article DOI: 10.1021/ml1000273 BindingDB Entry DOI: 10.7270/Q2FJ2H21
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Signal transducer and activator of transcription 3 (Homo sapiens (Human))	BDBM50338991 (CHEMBL1687979 \| N-[5-(2-Furyl)-1,3,4-oxadiazol-2-y...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	7.40E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Inhibition of STAT3 transcriptional activity in human HeLa cells by luciferase reporter gene assay				ACS Med Chem Lett 1: 371-375 (2010) Article DOI: 10.1021/ml1000273 BindingDB Entry DOI: 10.7270/Q2FJ2H21
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Signal transducer and activator of transcription 3 (Homo sapiens (Human))	BDBM50338997 (CHEMBL1687966 \| N-(5-Benzyl-1,3,4-oxadiazol-2-yl)-...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	7.50E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Inhibition of STAT3 transcriptional activity in human HeLa cells by luciferase reporter gene assay				ACS Med Chem Lett 1: 371-375 (2010) Article DOI: 10.1021/ml1000273 BindingDB Entry DOI: 10.7270/Q2FJ2H21
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Signal transducer and activator of transcription 3 (Homo sapiens (Human))	BDBM50338999 (2-Phenyl-N-[5-(2-thienyl)-1,3,4-oxadiazol-2-yl)-4-...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	7.50E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Inhibition of STAT3 transcriptional activity in human HeLa cells by luciferase reporter gene assay				ACS Med Chem Lett 1: 371-375 (2010) Article DOI: 10.1021/ml1000273 BindingDB Entry DOI: 10.7270/Q2FJ2H21
TBA Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%