Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Phospholipase A2 (Homo sapiens (Human)) | BDBM92676 (Manolide) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.30E+4 | n/a | n/a | n/a | n/a | 9.0 | 40 |
University of California, San Diego | Assay Description Inhibition assay using phospholipase A2. | J Biol Chem 264: 8520-8 (1989) BindingDB Entry DOI: 10.7270/Q2F76B48 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM92675 (7,7-dimethyl-5,8-eicosadienoic acid) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.60E+4 | n/a | n/a | n/a | n/a | 9.0 | 40 |
University of California, San Diego | Assay Description Inhibition assay using phospholipase A2. | J Biol Chem 264: 8520-8 (1989) BindingDB Entry DOI: 10.7270/Q2F76B48 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM92677 (Manoalogue) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.60E+4 | n/a | n/a | n/a | n/a | 9.0 | 40 |
University of California, San Diego | Assay Description Inhibition assay using phospholipase A2. | J Biol Chem 264: 8520-8 (1989) BindingDB Entry DOI: 10.7270/Q2F76B48 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM7876 (2-bromo-1-(4-bromophenyl)ethan-1-one | Halomethyl ...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid PDB UniChem Patents | PubMed | n/a | n/a | 5.50E+5 | n/a | n/a | n/a | n/a | 9.0 | 40 |
University of California, San Diego | Assay Description Inhibition assay using phospholipase A2. | J Biol Chem 264: 8520-8 (1989) BindingDB Entry DOI: 10.7270/Q2F76B48 | |||||||||||
More data for this Ligand-Target Pair |