Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Neuromedin-U receptor 2 (Homo sapiens (Human)) | BDBM50102660 (CHEBI:29081 | Oxedrine | Synephrine) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase DrugBank MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 6.60E+3 | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Agonist activity at human NMU2R transfected in HEK293 cells after 7 hrs by luciferase reporter gene assay | Bioorg Med Chem 22: 6117-23 (2014) Article DOI: 10.1016/j.bmc.2014.08.038 BindingDB Entry DOI: 10.7270/Q2XD13G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuromedin-U receptor 2 (Homo sapiens (Human)) | BDBM50217942 (2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4H-chr...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Agonist activity at human NMU2R transfected in HEK293 cells after 7 hrs by luciferase reporter gene assay | Bioorg Med Chem 22: 6117-23 (2014) Article DOI: 10.1016/j.bmc.2014.08.038 BindingDB Entry DOI: 10.7270/Q2XD13G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuromedin-U receptor 2 (Homo sapiens (Human)) | BDBM50102657 (CHEMBL3343016) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.53E+5 | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Agonist activity at human NMU2R transfected in HEK293 cells after 7 hrs by luciferase reporter gene assay | Bioorg Med Chem 22: 6117-23 (2014) Article DOI: 10.1016/j.bmc.2014.08.038 BindingDB Entry DOI: 10.7270/Q2XD13G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuromedin-U receptor 2 (Homo sapiens (Human)) | BDBM50102655 (CHEMBL3343014) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 7.30E+4 | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Agonist activity at human NMU2R transfected in HEK293 cells after 7 hrs by luciferase reporter gene assay | Bioorg Med Chem 22: 6117-23 (2014) Article DOI: 10.1016/j.bmc.2014.08.038 BindingDB Entry DOI: 10.7270/Q2XD13G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuromedin-U receptor 2 (Homo sapiens (Human)) | BDBM50102654 (CHEMBL3343013) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.11E+4 | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Agonist activity at human NMU2R transfected in HEK293 cells after 7 hrs by luciferase reporter gene assay | Bioorg Med Chem 22: 6117-23 (2014) Article DOI: 10.1016/j.bmc.2014.08.038 BindingDB Entry DOI: 10.7270/Q2XD13G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuromedin-U receptor 2 (Homo sapiens (Human)) | BDBM50102659 (CHEMBL3343023) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.70E+4 | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Agonist activity at human NMU2R transfected in HEK293 cells after 7 hrs by luciferase reporter gene assay | Bioorg Med Chem 22: 6117-23 (2014) Article DOI: 10.1016/j.bmc.2014.08.038 BindingDB Entry DOI: 10.7270/Q2XD13G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuromedin-U receptor 2 (Homo sapiens (Human)) | BDBM50049421 (CHEMBL3315349) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 6.10E+3 | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Agonist activity at human NMU2R transfected in HEK293 cells after 7 hrs by luciferase reporter gene assay | Bioorg Med Chem 22: 6117-23 (2014) Article DOI: 10.1016/j.bmc.2014.08.038 BindingDB Entry DOI: 10.7270/Q2XD13G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuromedin-U receptor 2 (Homo sapiens (Human)) | BDBM50102653 (CHEMBL3343012) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.73E+4 | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Agonist activity at human NMU2R transfected in HEK293 cells after 7 hrs by luciferase reporter gene assay | Bioorg Med Chem 22: 6117-23 (2014) Article DOI: 10.1016/j.bmc.2014.08.038 BindingDB Entry DOI: 10.7270/Q2XD13G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuromedin-U receptor 2 (Homo sapiens (Human)) | BDBM50102656 (CHEMBL3343015) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.40E+4 | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Agonist activity at human NMU2R transfected in HEK293 cells after 7 hrs by luciferase reporter gene assay | Bioorg Med Chem 22: 6117-23 (2014) Article DOI: 10.1016/j.bmc.2014.08.038 BindingDB Entry DOI: 10.7270/Q2XD13G1 | |||||||||||
More data for this Ligand-Target Pair |