Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cyclin-dependent kinase 1 (Homo sapiens (Human)) | BDBM50078891 (CHEMBL1973716) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Palermo Curated by ChEMBL | Assay Description Inhibition of CDC2 kinase (unknown origin) using histone H1 and [32P]-ATP | Eur J Med Chem 94: 149-62 (2015) Article DOI: 10.1016/j.ejmech.2015.03.005 BindingDB Entry DOI: 10.7270/Q2PG1TFS | |||||||||||
More data for this Ligand-Target Pair |