Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Casein kinase I isoform epsilon (Homo sapiens (Human)) | BDBM50082302 (CHEMBL3422700) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | 2.90E+4 | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" (IUBO-AG) Curated by ChEMBL | Assay Description Inhibition of human Casein kinase 1 epsilon | Eur J Med Chem 96: 308-17 (2015) Article DOI: 10.1016/j.ejmech.2015.03.046 BindingDB Entry DOI: 10.7270/Q2HD7XBQ | |||||||||||
More data for this Ligand-Target Pair |