Affinity Data by PubMed id=26003343

PubMed code 26003343

Found 10 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Estrogen receptor (Homo sapiens (Human))	BDBM50092526 (CHEMBL3586195) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.40	n/a	n/a	n/a	n/a	n/a	n/a
National Institute of Health Sciences Curated by ChEMBL					Assay Description Inhibition of ERalpha (unknown origin) by fluorescence polarization-based competition binding assay				Bioorg Med Chem 23: 3091-6 (2015) Article DOI: 10.1016/j.bmc.2015.05.002 BindingDB Entry DOI: 10.7270/Q28P6277
National Institute of Health Sciences Curated by ChEMBL					More data for this Ligand-Target Pair
Estrogen receptor (Homo sapiens (Human))	BDBM50092484 (CHEMBL3586191) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.60	n/a	n/a	n/a	n/a	n/a	n/a
National Institute of Health Sciences Curated by ChEMBL					Assay Description Inhibition of ERalpha (unknown origin) by fluorescence polarization-based competition binding assay				Bioorg Med Chem 23: 3091-6 (2015) Article DOI: 10.1016/j.bmc.2015.05.002 BindingDB Entry DOI: 10.7270/Q28P6277
National Institute of Health Sciences Curated by ChEMBL					More data for this Ligand-Target Pair
Estrogen receptor (Homo sapiens (Human))	BDBM50092523 (CHEMBL3586193) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.80	n/a	n/a	n/a	n/a	n/a	n/a
National Institute of Health Sciences Curated by ChEMBL					Assay Description Inhibition of ERalpha (unknown origin) by fluorescence polarization-based competition binding assay				Bioorg Med Chem 23: 3091-6 (2015) Article DOI: 10.1016/j.bmc.2015.05.002 BindingDB Entry DOI: 10.7270/Q28P6277
National Institute of Health Sciences Curated by ChEMBL					More data for this Ligand-Target Pair
Estrogen receptor (Homo sapiens (Human))	BDBM20608 (4-Hydroxytamoxifen \| 4-Hydroxytamoxifen (9) \| 4-[(...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	PDB Article PubMed	n/a	n/a	5.60	n/a	n/a	n/a	n/a	n/a	n/a
National Institute of Health Sciences Curated by ChEMBL					Assay Description Inhibition of ERalpha (unknown origin) by fluorescence polarization-based competition binding assay				Bioorg Med Chem 23: 3091-6 (2015) Article DOI: 10.1016/j.bmc.2015.05.002 BindingDB Entry DOI: 10.7270/Q28P6277
National Institute of Health Sciences Curated by ChEMBL					More data for this Ligand-Target Pair				3D Structure (crystal)
Estrogen receptor (Homo sapiens (Human))	BDBM50092522 (CHEMBL3586192) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	11	n/a	n/a	n/a	n/a	n/a	n/a
National Institute of Health Sciences Curated by ChEMBL					Assay Description Inhibition of ERalpha (unknown origin) by fluorescence polarization-based competition binding assay				Bioorg Med Chem 23: 3091-6 (2015) Article DOI: 10.1016/j.bmc.2015.05.002 BindingDB Entry DOI: 10.7270/Q28P6277
National Institute of Health Sciences Curated by ChEMBL					More data for this Ligand-Target Pair
Estrogen receptor (Homo sapiens (Human))	BDBM50092501 (CHEMBL3098274) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	14	n/a	n/a	n/a	n/a	n/a	n/a
National Institute of Health Sciences Curated by ChEMBL					Assay Description Inhibition of ERalpha (unknown origin) by fluorescence polarization-based competition binding assay				Bioorg Med Chem 23: 3091-6 (2015) Article DOI: 10.1016/j.bmc.2015.05.002 BindingDB Entry DOI: 10.7270/Q28P6277
National Institute of Health Sciences Curated by ChEMBL					More data for this Ligand-Target Pair
Estrogen receptor (Homo sapiens (Human))	BDBM50092483 (CHEMBL3586190) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	53	n/a	n/a	n/a	n/a	n/a	n/a
National Institute of Health Sciences Curated by ChEMBL					Assay Description Inhibition of ERalpha (unknown origin) by fluorescence polarization-based competition binding assay				Bioorg Med Chem 23: 3091-6 (2015) Article DOI: 10.1016/j.bmc.2015.05.002 BindingDB Entry DOI: 10.7270/Q28P6277
National Institute of Health Sciences Curated by ChEMBL					More data for this Ligand-Target Pair
Estrogen receptor (Homo sapiens (Human))	BDBM50092482 (CHEMBL3098273) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	151	n/a	n/a	n/a	n/a	n/a	n/a
National Institute of Health Sciences Curated by ChEMBL					Assay Description Inhibition of ERalpha (unknown origin) by fluorescence polarization-based competition binding assay				Bioorg Med Chem 23: 3091-6 (2015) Article DOI: 10.1016/j.bmc.2015.05.002 BindingDB Entry DOI: 10.7270/Q28P6277
National Institute of Health Sciences Curated by ChEMBL					More data for this Ligand-Target Pair
Estrogen receptor (Homo sapiens (Human))	BDBM50092525 (CHEMBL3586194) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	210	n/a	n/a	n/a	n/a	n/a	n/a
National Institute of Health Sciences Curated by ChEMBL					Assay Description Inhibition of ERalpha (unknown origin) by fluorescence polarization-based competition binding assay				Bioorg Med Chem 23: 3091-6 (2015) Article DOI: 10.1016/j.bmc.2015.05.002 BindingDB Entry DOI: 10.7270/Q28P6277
National Institute of Health Sciences Curated by ChEMBL					More data for this Ligand-Target Pair
Estrogen receptor (Homo sapiens (Human))	BDBM50092524 (CHEMBL3098275) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
National Institute of Health Sciences Curated by ChEMBL					Assay Description Inhibition of ERalpha (unknown origin) by fluorescence polarization-based competition binding assay				Bioorg Med Chem 23: 3091-6 (2015) Article DOI: 10.1016/j.bmc.2015.05.002 BindingDB Entry DOI: 10.7270/Q28P6277
National Institute of Health Sciences Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%