Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107287 (CHEMBL3601058) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.31E+4 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107315 (CHEMBL3601061) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.88E+4 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107304 (CHEMBL3601002) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 500 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107313 (CHEMBL3600994) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 160 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50107305 (CHEMBL3601001) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR41 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 2 (Homo sapiens (Human)) | BDBM50107303 (CHEMBL3601003) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR43 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107299 (CHEMBL3601007) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.13E+3 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107307 (CHEMBL3600999) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.75E+4 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 4 (Homo sapiens (Human)) | BDBM50107305 (CHEMBL3601001) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR120 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107306 (CHEMBL3601000) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 210 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107312 (CHEMBL3600995) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 560 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107286 (CHEMBL3601059) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.01E+4 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107292 (CHEMBL3601053) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.65E+3 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107298 (CHEMBL3601008) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107310 (CHEMBL3600997) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.07E+3 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50107303 (CHEMBL3601003) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR41 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107288 (CHEMBL3601057) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.58E+3 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107291 (CHEMBL3601054) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.67E+3 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107301 (CHEMBL3601005) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 680 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 2 (Homo sapiens (Human)) | BDBM50107305 (CHEMBL3601001) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR43 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 4 (Homo sapiens (Human)) | BDBM50107314 (CHEMBL3600993) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR120 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107290 (CHEMBL3601055) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107294 (CHEMBL3601051) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.39E+3 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107297 (CHEMBL3601049) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.26E+3 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107314 (CHEMBL3600993) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 58 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 4 (Homo sapiens (Human)) | BDBM50107303 (CHEMBL3601003) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR120 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107295 (CHEMBL3601050) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.12E+3 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107300 (CHEMBL3601006) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.11E+3 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107302 (CHEMBL3601004) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 610 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107303 (CHEMBL3601003) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 540 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107305 (CHEMBL3601001) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 300 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107309 (CHEMBL3600998) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.60E+3 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50107314 (CHEMBL3600993) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR41 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 2 (Homo sapiens (Human)) | BDBM50107314 (CHEMBL3600993) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR43 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107285 (CHEMBL3601060) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107293 (CHEMBL3601052) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.57E+3 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107311 (CHEMBL3600996) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 700 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 1 (Homo sapiens (Human)) | BDBM50107289 (CHEMBL3601056) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a |
Enamine Ltd Curated by ChEMBL | Assay Description Agonist activity at GPR40 (unknown origin) expressed in CHO cells by FLIPR calcium flux assay in presence of 0.1% bovine serum albumin | Bioorg Med Chem Lett 25: 3105-11 (2015) Article DOI: 10.1016/j.bmcl.2015.06.018 BindingDB Entry DOI: 10.7270/Q26D5VS5 | |||||||||||
More data for this Ligand-Target Pair |