Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Serine/threonine-protein kinase mTOR (Homo sapiens (Human)) | BDBM50103898 (CHEMBL3594042) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 613 | n/a | n/a | n/a | n/a | n/a | n/a |
India; Academy of Scientific and Innovative Research Curated by ChEMBL | Assay Description Inhibition of mTOR (unknown origin) assessed as p70S6K phosphorylation after 30 mins by ELISA | Bioorg Med Chem 23: 4237-47 (2015) Article DOI: 10.1016/j.bmc.2015.06.046 BindingDB Entry DOI: 10.7270/Q2D79D6T | |||||||||||
More data for this Ligand-Target Pair |