Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Polymerase acidic protein (Influenza A virus (strain A/X-31 H3N2)) | BDBM50122448 (CHEMBL463590 | L-742001) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 480 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Inhibition of recombinant Influenza virus A/X-31 N-terminal RdRp PA subunit (1 to 217) expressed in Escherichia coli using single-stranded circular D... | ACS Med Chem Lett 6: 866-71 (2015) Article DOI: 10.1021/acsmedchemlett.5b00109 BindingDB Entry DOI: 10.7270/Q27S7QKP | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Polymerase acidic protein (Influenza A virus (strain A/X-31 H3N2)) | BDBM50390688 (CHEMBL2070214) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 940 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Inhibition of recombinant Influenza virus A/X-31 N-terminal RdRp PA subunit (1 to 217) expressed in Escherichia coli using single-stranded circular D... | ACS Med Chem Lett 6: 866-71 (2015) Article DOI: 10.1021/acsmedchemlett.5b00109 BindingDB Entry DOI: 10.7270/Q27S7QKP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase acidic protein (Influenza A virus (strain A/X-31 H3N2)) | BDBM50122447 (CHEMBL3622460) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Inhibition of recombinant Influenza virus A/X-31 N-terminal RdRp PA subunit (1 to 217) expressed in Escherichia coli using single-stranded circular D... | ACS Med Chem Lett 6: 866-71 (2015) Article DOI: 10.1021/acsmedchemlett.5b00109 BindingDB Entry DOI: 10.7270/Q27S7QKP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase acidic protein (Influenza A virus (strain A/X-31 H3N2)) | BDBM50122443 (CHEMBL3622457) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Inhibition of recombinant Influenza virus A/X-31 N-terminal RdRp PA subunit (1 to 217) expressed in Escherichia coli using single-stranded circular D... | ACS Med Chem Lett 6: 866-71 (2015) Article DOI: 10.1021/acsmedchemlett.5b00109 BindingDB Entry DOI: 10.7270/Q27S7QKP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase acidic protein (Influenza A virus (strain A/X-31 H3N2)) | BDBM50122371 (CHEMBL3622452) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Inhibition of recombinant Influenza virus A/X-31 N-terminal RdRp PA subunit (1 to 217) expressed in Escherichia coli using single-stranded circular D... | ACS Med Chem Lett 6: 866-71 (2015) Article DOI: 10.1021/acsmedchemlett.5b00109 BindingDB Entry DOI: 10.7270/Q27S7QKP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase acidic protein (Influenza A virus (strain A/X-31 H3N2)) | BDBM50122438 (CHEMBL1611341) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Inhibition of recombinant Influenza virus A/X-31 N-terminal RdRp PA subunit (1 to 217) expressed in Escherichia coli using single-stranded circular D... | ACS Med Chem Lett 6: 866-71 (2015) Article DOI: 10.1021/acsmedchemlett.5b00109 BindingDB Entry DOI: 10.7270/Q27S7QKP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase acidic protein (Influenza A virus (strain A/X-31 H3N2)) | BDBM50122442 (CHEMBL3622456) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Inhibition of recombinant Influenza virus A/X-31 N-terminal RdRp PA subunit (1 to 217) expressed in Escherichia coli using single-stranded circular D... | ACS Med Chem Lett 6: 866-71 (2015) Article DOI: 10.1021/acsmedchemlett.5b00109 BindingDB Entry DOI: 10.7270/Q27S7QKP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase acidic protein (Influenza A virus (strain A/X-31 H3N2)) | BDBM50122445 (CHEMBL463072) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Inhibition of recombinant Influenza virus A/X-31 N-terminal RdRp PA subunit (1 to 217) expressed in Escherichia coli using single-stranded circular D... | ACS Med Chem Lett 6: 866-71 (2015) Article DOI: 10.1021/acsmedchemlett.5b00109 BindingDB Entry DOI: 10.7270/Q27S7QKP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase acidic protein (Influenza A virus (strain A/X-31 H3N2)) | BDBM50122446 (CHEMBL3622459) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Inhibition of recombinant Influenza virus A/X-31 N-terminal RdRp PA subunit (1 to 217) expressed in Escherichia coli using single-stranded circular D... | ACS Med Chem Lett 6: 866-71 (2015) Article DOI: 10.1021/acsmedchemlett.5b00109 BindingDB Entry DOI: 10.7270/Q27S7QKP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase acidic protein (Influenza A virus (strain A/X-31 H3N2)) | BDBM50122369 (CHEMBL3622450) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Inhibition of recombinant Influenza virus A/X-31 N-terminal RdRp PA subunit (1 to 217) expressed in Escherichia coli using single-stranded circular D... | ACS Med Chem Lett 6: 866-71 (2015) Article DOI: 10.1021/acsmedchemlett.5b00109 BindingDB Entry DOI: 10.7270/Q27S7QKP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase acidic protein (Influenza A virus (strain A/X-31 H3N2)) | BDBM50122370 (CHEMBL3622451) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Inhibition of recombinant Influenza virus A/X-31 N-terminal RdRp PA subunit (1 to 217) expressed in Escherichia coli using single-stranded circular D... | ACS Med Chem Lett 6: 866-71 (2015) Article DOI: 10.1021/acsmedchemlett.5b00109 BindingDB Entry DOI: 10.7270/Q27S7QKP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase acidic protein (Influenza A virus (strain A/X-31 H3N2)) | BDBM50122441 (CHEMBL3622455) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Inhibition of recombinant Influenza virus A/X-31 N-terminal RdRp PA subunit (1 to 217) expressed in Escherichia coli using single-stranded circular D... | ACS Med Chem Lett 6: 866-71 (2015) Article DOI: 10.1021/acsmedchemlett.5b00109 BindingDB Entry DOI: 10.7270/Q27S7QKP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase acidic protein (Influenza A virus (strain A/X-31 H3N2)) | BDBM50122444 (CHEMBL3622458) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Inhibition of recombinant Influenza virus A/X-31 N-terminal RdRp PA subunit (1 to 217) expressed in Escherichia coli using single-stranded circular D... | ACS Med Chem Lett 6: 866-71 (2015) Article DOI: 10.1021/acsmedchemlett.5b00109 BindingDB Entry DOI: 10.7270/Q27S7QKP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase acidic protein (Influenza A virus (strain A/X-31 H3N2)) | BDBM50122368 (CHEMBL3622449) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Inhibition of recombinant Influenza virus A/X-31 N-terminal RdRp PA subunit (1 to 217) expressed in Escherichia coli using single-stranded circular D... | ACS Med Chem Lett 6: 866-71 (2015) Article DOI: 10.1021/acsmedchemlett.5b00109 BindingDB Entry DOI: 10.7270/Q27S7QKP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase acidic protein (Influenza A virus (strain A/X-31 H3N2)) | BDBM50122440 (CHEMBL3622454) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Inhibition of recombinant Influenza virus A/X-31 N-terminal RdRp PA subunit (1 to 217) expressed in Escherichia coli using single-stranded circular D... | ACS Med Chem Lett 6: 866-71 (2015) Article DOI: 10.1021/acsmedchemlett.5b00109 BindingDB Entry DOI: 10.7270/Q27S7QKP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase acidic protein (Influenza A virus (strain A/X-31 H3N2)) | BDBM50122439 (CHEMBL3622453) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Sassari Curated by ChEMBL | Assay Description Inhibition of recombinant Influenza virus A/X-31 N-terminal RdRp PA subunit (1 to 217) expressed in Escherichia coli using single-stranded circular D... | ACS Med Chem Lett 6: 866-71 (2015) Article DOI: 10.1021/acsmedchemlett.5b00109 BindingDB Entry DOI: 10.7270/Q27S7QKP | |||||||||||
More data for this Ligand-Target Pair |