Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
DNA gyrase subunit A/B (Staphylococcus aureus) | BDBM50329257 (2-Hexadecynoic acid | CHEMBL1269411) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Inter American University of Puerto Rico Curated by ChEMBL | Assay Description Inhibition of supercoiling activity of Staphylococcus aureus DNA gyrase using relaxed pHOT1 plasmid DNA after 60 mins using ethidium bromide staining... | Bioorg Med Chem Lett 25: 5067-71 (2015) Article DOI: 10.1016/j.bmcl.2015.10.022 BindingDB Entry DOI: 10.7270/Q2GF0WBP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA gyrase subunit A/B (Staphylococcus aureus) | BDBM50133156 (CHEMBL3634703) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.26E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Inter American University of Puerto Rico Curated by ChEMBL | Assay Description Inhibition of supercoiling activity of Staphylococcus aureus DNA gyrase using relaxed pHOT1 plasmid DNA after 60 mins using ethidium bromide staining... | Bioorg Med Chem Lett 25: 5067-71 (2015) Article DOI: 10.1016/j.bmcl.2015.10.022 BindingDB Entry DOI: 10.7270/Q2GF0WBP | |||||||||||
More data for this Ligand-Target Pair |