Affinity Data by PubMed id=26682033

PubMed code 26682033

Found 30 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50430826 (CHEMBL2335155) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	199	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50430826 (CHEMBL2335155) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	200	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496778 (CHEMBL3220861) Show SMILES Cc1noc(C)c1-c1ccc2ncn(Cc3cccc(F)c3)c2c1 Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	631	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496772 (CHEMBL3220875) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	631	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496791 (CHEMBL3220869) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	631	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496787 (CHEMBL3220868) Show SMILES Cc1noc(C)c1-c1ccc2ncn(Cc3ccccc3Cl)c2c1 Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	794	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496792 (CHEMBL3220863) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	794	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496779 (CHEMBL3220867) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	794	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496780 (CHEMBL3220865) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496773 (CHEMBL3220871) Show SMILES Cc1noc(C)c1-c1ccc2ncn(Cc3ccccc3C#N)c2c1 Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496788 (CHEMBL3220874) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.26E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496793 (CHEMBL3220862) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.26E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496774 (CHEMBL3220860) Show SMILES Cc1noc(C)c1-c1ccc2CCC(O)(c2c1)c1ccccc1 Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid PDB UniChem	PDB Article PubMed	n/a	n/a	1.26E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair				3D Structure (crystal)
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496799 (CHEMBL3220850) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.59E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496781 (CHEMBL3220866) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.59E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496789 (CHEMBL3220876) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	2.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496798 (CHEMBL3220849) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	2.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496775 (CHEMBL3220864) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid PDB UniChem	Article PubMed	n/a	n/a	2.51E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496783 (CHEMBL3220859) Show SMILES Cc1noc(C)c1-c1ccc2CCC(OCCCN3CCNCC3)c2c1 Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	3.98E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496782 (CHEMBL3220872) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	3.98E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496776 (CHEMBL3220858) Show SMILES Cc1noc(C)c1-c1ccc2CCC(OCCCN3CCOCC3)c2c1 Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	6.31E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496784 (CHEMBL3220857) Show SMILES Cc1noc(C)c1-c1ccc2CCC(OCCCN3CCCCC3)c2c1 Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	6.31E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496785 (CHEMBL3220856) Show SMILES Cc1noc(C)c1-c1ccc2CCC(OCCCN3CCCC3)c2c1 Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	6.31E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496794 (CHEMBL3220853) Show SMILES Cc1noc(C)c1-c1ccc2nc[nH]c2c1 Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	6.31E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496790 (CHEMBL3220873) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496786 (CHEMBL3220870) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.26E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496796 (CHEMBL3220855) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	2.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496777 (CHEMBL3220852) Show SMILES Cc1noc(C)c1-c1ccc2cc[nH]c2c1 Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	2.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496797 (CHEMBL3220854) Show SMILES Cc1noc(C)c1-c1ccc2CCC(OCc3ccccc3)c2c1 Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	3.16E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Homo sapiens (Human))	BDBM50496795 (CHEMBL3220851) Show SMILES Cc1noc(C)c1-c1ccc2CCC(=O)c2c1 Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	6.31E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Oxford Curated by ChEMBL					Assay Description Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay				Medchemcomm 4: 140-144 (2013) Article DOI: 10.1039/c2md20189e BindingDB Entry DOI: 10.7270/Q2RX9G1D
University of Oxford Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%