Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Transcription activator BRG1 (Homo sapiens (Human)) | BDBM50266286 (CHEMBL4650213) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 263 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Oxford Curated by ChEMBL | Assay Description Alphascreen assay. Binding to SMARCA4A (domain start/stop: L1451-E1580) by alphascreen assay | Sci Adv 1: (2015) Article DOI: 10.1126/sciadv.1500723 BindingDB Entry DOI: 10.7270/Q2S75KX6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 (Homo sapiens (Human)) | BDBM50266286 (CHEMBL4650213) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 411 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Oxford Curated by ChEMBL | Assay Description Alphascreen assay. Binding to SMARCA4A (domain start/stop: L1451-E1580) by alphascreen assay | Sci Adv 1: (2015) Article DOI: 10.1126/sciadv.1500723 BindingDB Entry DOI: 10.7270/Q2S75KX6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein polybromo-1 (Homo sapiens (Human)) | BDBM50266286 (CHEMBL4650213) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 550 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Oxford Curated by ChEMBL | Assay Description Alphascreen assay. Binding to PB1A (domain start/stop: S613-D734) by alphascreen assay | Sci Adv 1: (2015) Article DOI: 10.1126/sciadv.1500723 BindingDB Entry DOI: 10.7270/Q2S75KX6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 (Homo sapiens (Human)) | BDBM50266286 (CHEMBL4650213) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 648 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Oxford Curated by ChEMBL | Assay Description Alphascreen assay. Binding to SMARCA4A (domain start/stop: L1451-E1580) by alphascreen assay | Sci Adv 1: (2015) Article DOI: 10.1126/sciadv.1500723 BindingDB Entry DOI: 10.7270/Q2S75KX6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein polybromo-1 (Homo sapiens (Human)) | BDBM50266286 (CHEMBL4650213) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 48 | n/a | n/a | n/a | n/a | n/a |
University of Oxford Curated by ChEMBL | Assay Description Reverse ITC (compound as receptor). Domain start/stop: S613-D734 | Sci Adv 1: (2015) Article DOI: 10.1126/sciadv.1500723 BindingDB Entry DOI: 10.7270/Q2S75KX6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 (Homo sapiens (Human)) | BDBM50266286 (CHEMBL4650213) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 89 | n/a | n/a | n/a | n/a | n/a |
University of Oxford Curated by ChEMBL | Assay Description Reverse ITC (compound as receptor). Domain start/stop: L1451-E1580 | Sci Adv 1: (2015) Article DOI: 10.1126/sciadv.1500723 BindingDB Entry DOI: 10.7270/Q2S75KX6 | |||||||||||
More data for this Ligand-Target Pair |