Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134635 (CHEMBL3746329 | US9637484, 3) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 34 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134637 (CHEMBL3746480 | US9637484, 2) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 61 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134675 (CHEMBL3747573 | US9637484, 22) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 115 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134634 (CHEMBL3745847 | US9637484, 31) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134670 (CHEMBL3745776 | US9637484, 7) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 159 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134644 (CHEMBL3746658 | US9637484, 9) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 198 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134645 (CHEMBL3746426 | US9637484, 5) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 207 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134677 (CHEMBL3747526 | US9637484, 32) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 324 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134672 (CHEMBL3747053) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 333 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134638 (CHEMBL3746315 | US9637484, 30) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 343 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134659 (CHEMBL3746049 | US9637484, 4) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 343 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134633 (CHEMBL3747024 | US9637484, 33) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 352 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134674 (CHEMBL3747747 | US9637484, 8) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 359 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134662 (CHEMBL3747493 | US9637484, 17) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 399 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134665 (CHEMBL3747343 | US9637484, 1) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 448 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134639 (CHEMBL3746433 | US9637484, 12) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 558 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134636 (CHEMBL3747353 | US9637484, 23) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 659 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134646 (CHEMBL3746317 | US9637484, 24) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 680 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134676 (CHEMBL3747094 | US9637484, 10) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 926 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134671 (CHEMBL3745813 | US9637484, 6) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.19E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134647 (CHEMBL3747215) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.26E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134673 (CHEMBL3747110) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.75E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134661 (CHEMBL3746048) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.79E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134643 (CHEMBL3747172) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.89E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134666 (CHEMBL3747643) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.93E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134658 (CHEMBL3746798) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.76E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134668 (CHEMBL3745763) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134664 (CHEMBL3747689) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134642 (CHEMBL3747474) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134660 (CHEMBL3746336) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134669 (CHEMBL3746459) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134641 (CHEMBL3746472) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134663 (CHEMBL3746789) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134667 (CHEMBL3747377) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 12 (Homo sapiens (Human)) | BDBM50134640 (CHEMBL3746178) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Hengrui Pharmaceutical Co. Ltd Curated by ChEMBL | Assay Description Inhibition of human URAT1 expressed in HEK293 cells assessed as [14C]uric acid uptake after 12 mins by scintillation counter | Bioorg Med Chem Lett 26: 277-82 (2016) Article DOI: 10.1016/j.bmcl.2015.12.040 BindingDB Entry DOI: 10.7270/Q2125VG4 | |||||||||||
More data for this Ligand-Target Pair |