Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Peroxisome proliferator-activated receptor alpha/delta/gamma (Homo sapiens (Human)) | BDBM50137094 (CHEMBL3754654) | PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.20E+4 | n/a | n/a | n/a | n/a |
Northwest A&F University Curated by ChEMBL | Assay Description Activation of PPAR (unknown origin) transactivation expressed in human HepG2 cells assessed as increase in transcriptional activity after 20 hrs by P... | Bioorg Med Chem Lett 26: 338-42 (2016) Article DOI: 10.1016/j.bmcl.2015.12.015 BindingDB Entry DOI: 10.7270/Q2QF8VQD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peroxisome proliferator-activated receptor alpha/delta/gamma (Homo sapiens (Human)) | BDBM50137095 (CHEMBL2335716) | PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.91E+4 | n/a | n/a | n/a | n/a |
Northwest A&F University Curated by ChEMBL | Assay Description Activation of PPAR (unknown origin) transactivation expressed in human HepG2 cells assessed as increase in transcriptional activity after 20 hrs by P... | Bioorg Med Chem Lett 26: 338-42 (2016) Article DOI: 10.1016/j.bmcl.2015.12.015 BindingDB Entry DOI: 10.7270/Q2QF8VQD | |||||||||||
More data for this Ligand-Target Pair |