Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Hepatocyte growth factor receptor (Homo sapiens (Human)) | BDBM50399540 (FORETINIB | US10464902, Foretinib | US10882853, Co...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE MMDB PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
Jiangxi Science& Technology Normal University Curated by ChEMBL | Assay Description Inhibition of c-Met (unknown origin) using FAM-labeled peptide substrate after 10 mins by mobility shift assay | Bioorg Med Chem 24: 1749-56 (2016) Article DOI: 10.1016/j.bmc.2016.02.046 BindingDB Entry DOI: 10.7270/Q2611258 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Hepatocyte growth factor receptor (Homo sapiens (Human)) | BDBM50154905 (CHEMBL3774821) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a |
Jiangxi Science& Technology Normal University Curated by ChEMBL | Assay Description Inhibition of c-Met (unknown origin) using FAM-labeled peptide substrate after 10 mins by mobility shift assay | Bioorg Med Chem 24: 1749-56 (2016) Article DOI: 10.1016/j.bmc.2016.02.046 BindingDB Entry DOI: 10.7270/Q2611258 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hepatocyte growth factor receptor (Homo sapiens (Human)) | BDBM50154908 (CHEMBL3775762) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 980 | n/a | n/a | n/a | n/a | n/a | n/a |
Jiangxi Science& Technology Normal University Curated by ChEMBL | Assay Description Inhibition of c-Met (unknown origin) using FAM-labeled peptide substrate after 10 mins by mobility shift assay | Bioorg Med Chem 24: 1749-56 (2016) Article DOI: 10.1016/j.bmc.2016.02.046 BindingDB Entry DOI: 10.7270/Q2611258 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hepatocyte growth factor receptor (Homo sapiens (Human)) | BDBM50154907 (CHEMBL3775533) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Jiangxi Science& Technology Normal University Curated by ChEMBL | Assay Description Inhibition of c-Met (unknown origin) using FAM-labeled peptide substrate after 10 mins by mobility shift assay | Bioorg Med Chem 24: 1749-56 (2016) Article DOI: 10.1016/j.bmc.2016.02.046 BindingDB Entry DOI: 10.7270/Q2611258 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Hepatocyte growth factor receptor (Homo sapiens (Human)) | BDBM50154906 (CHEMBL3775074) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Jiangxi Science& Technology Normal University Curated by ChEMBL | Assay Description Inhibition of c-Met (unknown origin) using FAM-labeled peptide substrate after 10 mins by mobility shift assay | Bioorg Med Chem 24: 1749-56 (2016) Article DOI: 10.1016/j.bmc.2016.02.046 BindingDB Entry DOI: 10.7270/Q2611258 | |||||||||||
More data for this Ligand-Target Pair |