Affinity Data by PubMed id=26974383

PubMed code 26974383

Found 11 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Amine oxidase [flavin-containing] B (Homo sapiens (Human))	BDBM50155318 (CHEMBL3781063) Show SMILES CSc1ccc(cc1)C(=O)\C=C\c1cccc2OCOc12 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	550	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Qatar University Curated by ChEMBL					Assay Description Competitive inhibition of human MAOB overexpressed in Pichia pastoris using MMTP as substrate preincubated for 5 mins followed by substrate addition ...				Eur J Med Chem 114: 162-9 (2016) Article DOI: 10.1016/j.ejmech.2016.02.038 BindingDB Entry DOI: 10.7270/Q2N018F1
Qatar University Curated by ChEMBL					More data for this Ligand-Target Pair
Amine oxidase [flavin-containing] B (Homo sapiens (Human))	BDBM50155319 (CHEMBL3781774) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	720	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Qatar University Curated by ChEMBL					Assay Description Competitive inhibition of human MAOB overexpressed in Pichia pastoris using MMTP as substrate preincubated for 5 mins followed by substrate addition ...				Eur J Med Chem 114: 162-9 (2016) Article DOI: 10.1016/j.ejmech.2016.02.038 BindingDB Entry DOI: 10.7270/Q2N018F1
Qatar University Curated by ChEMBL					More data for this Ligand-Target Pair
Amine oxidase [flavin-containing] B (Homo sapiens (Human))	BDBM50155322 (CHEMBL3780640) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	780	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Qatar University Curated by ChEMBL					Assay Description Competitive inhibition of human MAOB overexpressed in Pichia pastoris using MMTP as substrate preincubated for 5 mins followed by substrate addition ...				Eur J Med Chem 114: 162-9 (2016) Article DOI: 10.1016/j.ejmech.2016.02.038 BindingDB Entry DOI: 10.7270/Q2N018F1
Qatar University Curated by ChEMBL					More data for this Ligand-Target Pair
Amine oxidase [flavin-containing] B (Homo sapiens (Human))	BDBM50155321 (CHEMBL3782038) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	1.15E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Qatar University Curated by ChEMBL					Assay Description Competitive inhibition of human MAOB overexpressed in Pichia pastoris using MMTP as substrate preincubated for 5 mins followed by substrate addition ...				Eur J Med Chem 114: 162-9 (2016) Article DOI: 10.1016/j.ejmech.2016.02.038 BindingDB Entry DOI: 10.7270/Q2N018F1
Qatar University Curated by ChEMBL					More data for this Ligand-Target Pair
Amine oxidase [flavin-containing] B (Homo sapiens (Human))	BDBM50155312 (CHEMBL3780160) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	2.36E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Qatar University Curated by ChEMBL					Assay Description Competitive inhibition of human MAOB overexpressed in Pichia pastoris using MMTP as substrate preincubated for 5 mins followed by substrate addition ...				Eur J Med Chem 114: 162-9 (2016) Article DOI: 10.1016/j.ejmech.2016.02.038 BindingDB Entry DOI: 10.7270/Q2N018F1
Qatar University Curated by ChEMBL					More data for this Ligand-Target Pair
Amine oxidase [flavin-containing] B (Homo sapiens (Human))	BDBM50155322 (CHEMBL3780640) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	n/a
Qatar University Curated by ChEMBL					Assay Description Inhibition of recombinant human MAOB expressed in baculovirus infected BTI insect cell microsomes using MMTP as substrate preincubated for 5 mins fol...				Eur J Med Chem 114: 162-9 (2016) Article DOI: 10.1016/j.ejmech.2016.02.038 BindingDB Entry DOI: 10.7270/Q2N018F1
Qatar University Curated by ChEMBL					More data for this Ligand-Target Pair
Amine oxidase [flavin-containing] B (Homo sapiens (Human))	BDBM50155318 (CHEMBL3781063) Show SMILES CSc1ccc(cc1)C(=O)\C=C\c1cccc2OCOc12 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	950	n/a	n/a	n/a	n/a	n/a	n/a
Qatar University Curated by ChEMBL					Assay Description Inhibition of recombinant human MAOB expressed in baculovirus infected BTI insect cell microsomes using MMTP as substrate preincubated for 5 mins fol...				Eur J Med Chem 114: 162-9 (2016) Article DOI: 10.1016/j.ejmech.2016.02.038 BindingDB Entry DOI: 10.7270/Q2N018F1
Qatar University Curated by ChEMBL					More data for this Ligand-Target Pair
Amine oxidase [flavin-containing] B (Homo sapiens (Human))	BDBM50155319 (CHEMBL3781774) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Qatar University Curated by ChEMBL					Assay Description Inhibition of recombinant human MAOB expressed in baculovirus infected BTI insect cell microsomes using MMTP as substrate preincubated for 5 mins fol...				Eur J Med Chem 114: 162-9 (2016) Article DOI: 10.1016/j.ejmech.2016.02.038 BindingDB Entry DOI: 10.7270/Q2N018F1
Qatar University Curated by ChEMBL					More data for this Ligand-Target Pair
Amine oxidase [flavin-containing] B (Homo sapiens (Human))	BDBM50155312 (CHEMBL3780160) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.51E+3	n/a	n/a	n/a	n/a	n/a	n/a
Qatar University Curated by ChEMBL					Assay Description Inhibition of recombinant human MAOB expressed in baculovirus infected BTI insect cell microsomes using MMTP as substrate preincubated for 5 mins fol...				Eur J Med Chem 114: 162-9 (2016) Article DOI: 10.1016/j.ejmech.2016.02.038 BindingDB Entry DOI: 10.7270/Q2N018F1
Qatar University Curated by ChEMBL					More data for this Ligand-Target Pair
Amine oxidase [flavin-containing] B (Homo sapiens (Human))	BDBM50155321 (CHEMBL3782038) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.97E+3	n/a	n/a	n/a	n/a	n/a	n/a
Qatar University Curated by ChEMBL					Assay Description Inhibition of recombinant human MAOB expressed in baculovirus infected BTI insect cell microsomes using MMTP as substrate preincubated for 5 mins fol...				Eur J Med Chem 114: 162-9 (2016) Article DOI: 10.1016/j.ejmech.2016.02.038 BindingDB Entry DOI: 10.7270/Q2N018F1
Qatar University Curated by ChEMBL					More data for this Ligand-Target Pair
Amine oxidase [flavin-containing] B (Homo sapiens (Human))	BDBM50155320 (CHEMBL3781364) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	4.49E+3	n/a	n/a	n/a	n/a	n/a	n/a
Qatar University Curated by ChEMBL					Assay Description Inhibition of recombinant human MAOB expressed in baculovirus infected BTI insect cell microsomes using MMTP as substrate preincubated for 5 mins fol...				Eur J Med Chem 114: 162-9 (2016) Article DOI: 10.1016/j.ejmech.2016.02.038 BindingDB Entry DOI: 10.7270/Q2N018F1
Qatar University Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%