Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50156812 (PHENSTATIN) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
'Al. I. Cuza' University of Iasi Curated by ChEMBL | Assay Description Inhibition of bovine tubulin polymerization preincubated for 30 mins followed by GTP addition measured after 20 mins by spectrophotometric method | Bioorg Med Chem 24: 2307-17 (2016) Article DOI: 10.1016/j.bmc.2016.04.001 BindingDB Entry DOI: 10.7270/Q2KW5HX2 | |||||||||||
More data for this Ligand-Target Pair |