Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50536020 (CHEMBL4464873) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Chicago State University Curated by ChEMBL | Assay Description Inhibition of human ERG | J Med Chem 59: 6232-47 (2016) Article DOI: 10.1021/acs.jmedchem.6b00415 BindingDB Entry DOI: 10.7270/Q2DB85CT | |||||||||||
More data for this Ligand-Target Pair |