Found 25 hits of Enzyme Inhibition Constant Data Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50234336
(CHEMBL4093667)Show SMILES OC(=O)c1ccc(-c2c[nH]c3ncc(cc23)-c2ccccc2)c(F)c1 Show InChI InChI=1S/C20H13FN2O2/c21-18-9-13(20(24)25)6-7-15(18)17-11-23-19-16(17)8-14(10-22-19)12-4-2-1-3-5-12/h1-11H,(H,22,23)(H,24,25) | PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet 
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 111 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50234329
(CHEMBL4083405)Show SMILES OC(=O)c1ccc(cc1F)-c1c[nH]c2ncc(cc12)-c1ccccc1 Show InChI InChI=1S/C20H13FN2O2/c21-18-9-13(6-7-15(18)20(24)25)17-11-23-19-16(17)8-14(10-22-19)12-4-2-1-3-5-12/h1-11H,(H,22,23)(H,24,25) | PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 118 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50296003
(4-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl)benzoic ...)Show SMILES OC(=O)c1ccc(cc1)-c1c[nH]c2ncc(cc12)-c1ccccc1 Show InChI InChI=1S/C20H14N2O2/c23-20(24)15-8-6-14(7-9-15)18-12-22-19-17(18)10-16(11-21-19)13-4-2-1-3-5-13/h1-12H,(H,21,22)(H,23,24) | PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
DrugBank
MMDB
PC cid
PC sid
PDB
UniChem
Patents
Similars
| Article
PubMed
| n/a | n/a | 182 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50234330
(CHEMBL4101393)Show SMILES OC(=O)c1cc(F)cc(c1)-c1c[nH]c2ncc(cc12)-c1ccccc1 Show InChI InChI=1S/C20H13FN2O2/c21-16-7-13(6-14(8-16)20(24)25)18-11-23-19-17(18)9-15(10-22-19)12-4-2-1-3-5-12/h1-11H,(H,22,23)(H,24,25) | PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| Article
PubMed
| n/a | n/a | 340 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50296008
(3-(4-(1H-tetrazol-5-yl)phenyl)-5-phenyl-1H-pyrrolo...)Show SMILES c1[nH]c2ncc(cc2c1-c1ccc(cc1)-c1nnn[nH]1)-c1ccccc1 Show InChI InChI=1S/C20H14N6/c1-2-4-13(5-3-1)16-10-17-18(12-22-20(17)21-11-16)14-6-8-15(9-7-14)19-23-25-26-24-19/h1-12H,(H,21,22)(H,23,24,25,26) | PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
| Article
PubMed
| n/a | n/a | 524 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50234326
(CHEMBL4102305)Show SMILES OC(=O)c1cccc(c1)-c1c[nH]c2ncc(cc12)-c1ccccc1 Show InChI InChI=1S/C20H14N2O2/c23-20(24)15-8-4-7-14(9-15)18-12-22-19-17(18)10-16(11-21-19)13-5-2-1-3-6-13/h1-12H,(H,21,22)(H,23,24) | PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| Article
PubMed
| n/a | n/a | 896 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50234337
(CHEMBL4102893)Show SMILES OC(=O)c1cc(ccc1F)-c1c[nH]c2ncc(cc12)-c1ccccc1 Show InChI InChI=1S/C20H13FN2O2/c21-18-7-6-13(8-16(18)20(24)25)17-11-23-19-15(17)9-14(10-22-19)12-4-2-1-3-5-12/h1-11H,(H,22,23)(H,24,25) | PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| Article
PubMed
| n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50234332
(CHEMBL4079544)Show InChI InChI=1S/C15H12N2O2/c1-19-15(18)13-9-17-14-12(13)7-11(8-16-14)10-5-3-2-4-6-10/h2-9H,1H3,(H,16,17) | PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
| Article
PubMed
| n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50234320
(CHEMBL4103803)Show InChI InChI=1S/C14H11N3O2/c1-19-14(18)12-8-17-13-11(12)6-10(7-16-13)9-2-4-15-5-3-9/h2-8H,1H3,(H,16,17) | PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50234328
(CHEMBL4072966)Show SMILES OC(=O)c1ccc(cc1)-c1cnc2[nH]cc(-c3ccccc3)c2c1 Show InChI InChI=1S/C20H14N2O2/c23-20(24)15-8-6-13(7-9-15)16-10-17-18(12-22-19(17)21-11-16)14-4-2-1-3-5-14/h1-12H,(H,21,22)(H,23,24) | PDB
KEGG
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B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 1.94E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50234322
(CHEMBL4096050)Show InChI InChI=1S/C13H10N2O2S/c1-17-13(16)11-6-15-12-10(11)4-9(5-14-12)8-2-3-18-7-8/h2-7H,1H3,(H,14,15) | PDB
KEGG
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antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 2.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50234321
(CHEMBL4068740)Show InChI InChI=1S/C14H11N3O2/c1-19-14(18)11-8-17-13-10(11)6-9(7-16-13)12-4-2-3-5-15-12/h2-8H,1H3,(H,16,17) | PDB
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GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 2.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50234325
(CHEMBL4092680)Show InChI InChI=1S/C20H14N2O/c23-13-14-5-4-8-16(9-14)19-12-22-20-18(19)10-17(11-21-20)15-6-2-1-3-7-15/h1-13H,(H,21,22) | PDB
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| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 3.45E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50445250
(CHEMBL3102859)Show InChI InChI=1S/C19H14N2/c1-3-7-14(8-4-1)16-11-17-18(13-21-19(17)20-12-16)15-9-5-2-6-10-15/h1-13H,(H,20,21) | PDB
KEGG
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GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 4.06E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50234333
(CHEMBL4095116)Show InChI InChI=1S/C13H10N2O3/c1-17-13(16)10-7-15-12-9(10)5-8(6-14-12)11-3-2-4-18-11/h2-7H,1H3,(H,14,15) | PDB
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GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
| Article
PubMed
| n/a | n/a | 6.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50234317
(CHEMBL4090019)Show InChI InChI=1S/C13H10N4O/c18-13(17-9-3-1-5-14-7-9)11-8-16-12-10(11)4-2-6-15-12/h1-8H,(H,15,16)(H,17,18) | PDB
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GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50234335
(CHEMBL4066045)Show InChI InChI=1S/C19H16N4/c1-2-5-14(6-3-1)15-9-18-16(12-23-19(18)22-10-15)11-21-17-7-4-8-20-13-17/h1-10,12-13,21H,11H2,(H,22,23) | PDB
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| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50234323
(CHEMBL4087427)Show InChI InChI=1S/C20H15N3O/c24-20(23-16-9-5-2-6-10-16)18-13-22-19-17(18)11-15(12-21-19)14-7-3-1-4-8-14/h1-13H,(H,21,22)(H,23,24) | PDB
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PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50234319
(CHEMBL4100172)Show InChI InChI=1S/C14H11N3O2/c1-19-14(18)12-7-10-6-11(8-16-13(10)17-12)9-2-4-15-5-3-9/h2-8H,1H3,(H,16,17) | PDB
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| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50234316
(CHEMBL2391621)Show InChI InChI=1S/C9H8N2O2/c1-13-9(12)7-5-11-8-6(7)3-2-4-10-8/h2-5H,1H3,(H,10,11) | PDB
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CHEMBL
MCE
PC cid
PC sid
PDB
UniChem
Similars
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50234318
(CHEMBL4091294)Show InChI InChI=1S/C13H10N2/c1-2-4-10(5-3-1)12-8-11-6-7-14-13(11)15-9-12/h1-9H,(H,14,15) | PDB
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CHEMBL
PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50234315
(CHEMBL4097745)Show InChI InChI=1S/C9H8N2O2/c1-13-9(12)7-5-6-3-2-4-10-8(6)11-7/h2-5H,1H3,(H,10,11) | PDB
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CHEMBL
MCE
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50234324
(CHEMBL4064994)Show SMILES COC(=O)c1cccc(c1)-c1c[nH]c2ncc(cc12)-c1ccccc1 Show InChI InChI=1S/C21H16N2O2/c1-25-21(24)16-9-5-8-15(10-16)19-13-23-20-18(19)11-17(12-22-20)14-6-3-2-4-7-14/h2-13H,1H3,(H,22,23) | PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50234331
(CHEMBL4061976)Show InChI InChI=1S/C11H9N5O/c17-11(15-9-3-5-14-16-9)8-6-13-10-7(8)2-1-4-12-10/h1-6H,(H,12,13)(H2,14,15,16,17) | PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human)) | BDBM50234327
(CHEMBL4085916)Show SMILES OC(=O)c1cccc(c1)-c1cnc2[nH]cc(-c3ccccc3)c2c1 Show InChI InChI=1S/C20H14N2O2/c23-20(24)15-8-4-7-14(9-15)16-10-17-18(12-22-19(17)21-11-16)13-5-2-1-3-6-13/h1-12H,(H,21,22)(H,23,24) | PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 1.02E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
OriBase Pharma
Curated by ChEMBL
| Assay Description
Inhibition of recombinant human His-tagged AXL expressed in insect cells after 60 mins by Z'-LYTE assay |
Bioorg Med Chem Lett 27: 862-866 (2017)
Article DOI: 10.1016/j.bmcl.2017.01.015
BindingDB Entry DOI: 10.7270/Q24M96S8 |
More data for this
Ligand-Target Pair | |
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