Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Transthyretin (Homo sapiens (Human)) | BDBM50249584 (CHEMBL4074607) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a |
CIC bioGUNE , Bizkaia Technology Park, Building 801A, 48170 Derio, Spain. Curated by ChEMBL | Assay Description Binding affinity to recombinant human transthyretin expressed in Escherichia coli BL21 by STD-NMR spectroscopic method | J Med Chem 60: 5749-5758 (2017) Article DOI: 10.1021/acs.jmedchem.7b00428 BindingDB Entry DOI: 10.7270/Q29W0HW7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transthyretin (Homo sapiens (Human)) | BDBM50070942 ((-)-Epigallocatechin gallate | (-)-Epigallocatechi...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG MMDB PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a |
CIC bioGUNE , Bizkaia Technology Park, Building 801A, 48170 Derio, Spain. Curated by ChEMBL | Assay Description Binding affinity to recombinant human transthyretin expressed in Escherichia coli BL21 by STD-NMR spectroscopic method | J Med Chem 60: 5749-5758 (2017) Article DOI: 10.1021/acs.jmedchem.7b00428 BindingDB Entry DOI: 10.7270/Q29W0HW7 | |||||||||||
More data for this Ligand-Target Pair |