Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Tyrosyl-DNA phosphodiesterase 1 (Homo sapiens (Human)) | BDBM50269845 (CHEMBL4077630) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Griffith Institute for Drug Discovery, Griffith University, Brisbane QLD 4111, Australia. Curated by ChEMBL | Assay Description Inhibition of Tdp1 (unknown origin) using 5'-(6-TAMN-AGGATCTAAAAGACTT-BHQ-)3' as substrate pretreated for 30 mins followed by substrate addition by f... | Bioorg Med Chem Lett 27: 4007-4010 (2017) Article DOI: 10.1016/j.bmcl.2017.07.062 BindingDB Entry DOI: 10.7270/Q2765HTQ | |||||||||||
More data for this Ligand-Target Pair |