Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50242191 (CHEMBL4083511) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Crystal Pharmatech Co., Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit the activity of K+ stimulated gastric ATPase | J Med Chem 60: 8847-8857 (2017) Article DOI: 10.1021/acs.jmedchem.7b00971 BindingDB Entry DOI: 10.7270/Q2QV3PWT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM217379 (CDDO-Me, 2) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | >2.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Crystal Pharmatech Co., Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit the activity of K+ stimulated gastric ATPase | J Med Chem 60: 8847-8857 (2017) Article DOI: 10.1021/acs.jmedchem.7b00971 BindingDB Entry DOI: 10.7270/Q2QV3PWT | |||||||||||
More data for this Ligand-Target Pair |