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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50773 (1-[4-(2-methoxyphenyl)-1-piperazinyl]-3-(1-naphtha...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet  | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Guangzhou Medical University Curated by ChEMBL | Assay Description Displacement of [125I-HEAT from human alpha1D-adrenoreceptor expressed in CHOK1 cell membranes incubated for 60 mins | Bioorg Med Chem Lett 28: 547-551 (2018) Article DOI: 10.1016/j.bmcl.2018.01.068 BindingDB Entry DOI: 10.7270/Q2057JHB | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50773 (1-[4-(2-methoxyphenyl)-1-piperazinyl]-3-(1-naphtha...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 3.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Guangzhou Medical University Curated by ChEMBL | Assay Description Displacement of [125I-HEAT from human alpha1A-adrenoreceptor expressed in CHOK1 cell membranes incubated for 60 mins | Bioorg Med Chem Lett 28: 547-551 (2018) Article DOI: 10.1016/j.bmcl.2018.01.068 BindingDB Entry DOI: 10.7270/Q2057JHB | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50773 (1-[4-(2-methoxyphenyl)-1-piperazinyl]-3-(1-naphtha...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Guangzhou Medical University Curated by ChEMBL | Assay Description Displacement of [125I-HEAT from human alpha1B-adrenoreceptor expressed in CHOK1 cell membranes incubated for 60 mins | Bioorg Med Chem Lett 28: 547-551 (2018) Article DOI: 10.1016/j.bmcl.2018.01.068 BindingDB Entry DOI: 10.7270/Q2057JHB | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
