Affinity Data by PubMed id=3005567

PubMed code 3005567

Found 7 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Sodium- and chloride-dependent betaine transporter (Rattus norvegicus)	BDBM50226144 (2,4-Diamino-Butyric Acid \| CHEBI:64307 \| CHEMBL307...) Show SMILES NCCC(N)C(O)=O Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	2.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.				J Med Chem 29: 224-9 (1986) BindingDB Entry DOI: 10.7270/Q2FX7CNP
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent betaine transporter (Rattus norvegicus)	BDBM50226141 (CHEMBL309688) Show SMILES Oc1onc2CCNCc12 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	1.30E+5	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.				J Med Chem 29: 224-9 (1986) BindingDB Entry DOI: 10.7270/Q2FX7CNP
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent betaine transporter (Rattus norvegicus)	BDBM50226145 (CHEMBL150830) Show SMILES Oc1noc2CCNCc12 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	1.60E+5	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.				J Med Chem 29: 224-9 (1986) BindingDB Entry DOI: 10.7270/Q2FX7CNP
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent betaine transporter (Rattus norvegicus)	BDBM50224808 (CHEMBL309689) Show SMILES Oc1noc2CCNCCc12 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.				J Med Chem 29: 224-9 (1986) BindingDB Entry DOI: 10.7270/Q2FX7CNP
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent betaine transporter (Rattus norvegicus)	BDBM50226143 (CHEMBL305673) Show SMILES Oc1onc2CCCNCc12 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.				J Med Chem 29: 224-9 (1986) BindingDB Entry DOI: 10.7270/Q2FX7CNP
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent betaine transporter (Rattus norvegicus)	BDBM50226146 (CHEMBL74364) Show SMILES Oc1onc2CNCCCc12 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.				J Med Chem 29: 224-9 (1986) BindingDB Entry DOI: 10.7270/Q2FX7CNP
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium- and chloride-dependent betaine transporter (Rattus norvegicus)	BDBM50226142 (CHEMBL292757) Show SMILES Oc1onc2CCNCCc12 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.				J Med Chem 29: 224-9 (1986) BindingDB Entry DOI: 10.7270/Q2FX7CNP
TBA Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%