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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Metabotropic glutamate receptor 2 (Rattus norvegicus) | BDBM50559786 (CHEMBL4800093) | PDB UniProtKB/SwissProt GoogleScholar AffyNet  | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 54 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulation of rat mGlu2 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127212 BindingDB Entry DOI: 10.7270/Q27H1P86 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Metabotropic glutamate receptor 4 (Rattus norvegicus (Rat)) | BDBM50559791 (CHEMBL4740929) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 32 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulation of rat mGlu4 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127212 BindingDB Entry DOI: 10.7270/Q27H1P86 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Metabotropic glutamate receptor 2 (Rattus norvegicus) | BDBM50559794 (CHEMBL4752318) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 69 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulation of rat mGlu2 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127212 BindingDB Entry DOI: 10.7270/Q27H1P86 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Metabotropic glutamate receptor 2 (Rattus norvegicus) | BDBM50559787 (CHEMBL4786847) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 98 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulation of rat mGlu2 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127212 BindingDB Entry DOI: 10.7270/Q27H1P86 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Metabotropic glutamate receptor 2 (Rattus norvegicus) | BDBM50559790 (CHEMBL4744407) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 122 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulation of rat mGlu2 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127212 BindingDB Entry DOI: 10.7270/Q27H1P86 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Metabotropic glutamate receptor 2 (Rattus norvegicus) | BDBM50559792 (CHEMBL4759458) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 134 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulation of rat mGlu2 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127212 BindingDB Entry DOI: 10.7270/Q27H1P86 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Metabotropic glutamate receptor 4 (Rattus norvegicus (Rat)) | BDBM50559785 (CHEMBL4748549) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 657 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulation of rat mGlu4 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127212 BindingDB Entry DOI: 10.7270/Q27H1P86 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Metabotropic glutamate receptor 2 (Rattus norvegicus) | BDBM50559785 (CHEMBL4748549) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 281 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulation of rat mGlu2 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127212 BindingDB Entry DOI: 10.7270/Q27H1P86 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Metabotropic glutamate receptor 4 (Rattus norvegicus (Rat)) | BDBM50559787 (CHEMBL4786847) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 33 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulation of rat mGlu4 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127212 BindingDB Entry DOI: 10.7270/Q27H1P86 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Metabotropic glutamate receptor 4 (Rattus norvegicus (Rat)) | BDBM55082 (N-[4-[(2-chlorobenzoyl)amino]-3-methoxy-phenyl]pic...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 34 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulation of rat mGlu4 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127212 BindingDB Entry DOI: 10.7270/Q27H1P86 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Metabotropic glutamate receptor 4 (Rattus norvegicus (Rat)) | BDBM50559786 (CHEMBL4800093) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 38 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulation of rat mGlu4 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127212 BindingDB Entry DOI: 10.7270/Q27H1P86 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Metabotropic glutamate receptor 2 (Rattus norvegicus) | BDBM50559789 (CHEMBL4762369) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 62 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulation of rat mGlu2 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127212 BindingDB Entry DOI: 10.7270/Q27H1P86 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Metabotropic glutamate receptor 2 (Rattus norvegicus) | BDBM50559793 (CHEMBL4748285) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.18E+3 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulation of rat mGlu2 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127212 BindingDB Entry DOI: 10.7270/Q27H1P86 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Metabotropic glutamate receptor 2 (Rattus norvegicus) | BDBM50559795 (CHEMBL4779278) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 62 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulation of rat mGlu2 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127212 BindingDB Entry DOI: 10.7270/Q27H1P86 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Metabotropic glutamate receptor 4 (Rattus norvegicus (Rat)) | BDBM50559788 (CHEMBL4777845) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 35 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulation of rat mGlu4 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127212 BindingDB Entry DOI: 10.7270/Q27H1P86 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Metabotropic glutamate receptor 4 (Rattus norvegicus (Rat)) | BDBM50559790 (CHEMBL4744407) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 30 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulation of rat mGlu4 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127212 BindingDB Entry DOI: 10.7270/Q27H1P86 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Metabotropic glutamate receptor 4 (Rattus norvegicus (Rat)) | BDBM50559792 (CHEMBL4759458) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulation of rat mGlu4 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127212 BindingDB Entry DOI: 10.7270/Q27H1P86 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Metabotropic glutamate receptor 4 (Rattus norvegicus (Rat)) | BDBM50559793 (CHEMBL4748285) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulation of rat mGlu4 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127212 BindingDB Entry DOI: 10.7270/Q27H1P86 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Metabotropic glutamate receptor 2 (Rattus norvegicus) | BDBM50559784 (CHEMBL4761801) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 84 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulation of rat mGlu2 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127212 BindingDB Entry DOI: 10.7270/Q27H1P86 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Metabotropic glutamate receptor 2 (Rattus norvegicus) | BDBM50559788 (CHEMBL4777845) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 92 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulation of rat mGlu2 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127212 BindingDB Entry DOI: 10.7270/Q27H1P86 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Metabotropic glutamate receptor 4 (Rattus norvegicus (Rat)) | BDBM50559789 (CHEMBL4762369) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 32 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulation of rat mGlu4 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127212 BindingDB Entry DOI: 10.7270/Q27H1P86 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Metabotropic glutamate receptor 2 (Rattus norvegicus) | BDBM50559791 (CHEMBL4740929) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 94 | n/a | n/a | n/a | n/a |
TBA | Assay Description Positive allosteric modulation of rat mGlu2 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127212 BindingDB Entry DOI: 10.7270/Q27H1P86 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
