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Articleid 50030082

Compile data set for download or QSAR
Found 56 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Endothelin-1 receptor


(RAT)		BDBM50290940
PNG
(CHEMBL94929 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3,5-di...)
Show SMILES Cc1cc(C)c(=O)n(n1)C(C(=O)NS(=O)(=O)c1ccc(cc1)C(C)(C)C)c1ccc2OCOc2c1
Show InChI InChI=1S/C25H27N3O6S/c1-15-12-16(2)26-28(24(15)30)22(17-6-11-20-21(13-17)34-14-33-20)23(29)27-35(31,32)19-9-7-18(8-10-19)25(3,4)5/h6-13,22H,14H2,1-5H3,(H,27,29)
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n/an/a 18n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290940
PNG
(CHEMBL94929 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3,5-di...)
Show SMILES Cc1cc(C)c(=O)n(n1)C(C(=O)NS(=O)(=O)c1ccc(cc1)C(C)(C)C)c1ccc2OCOc2c1
Show InChI InChI=1S/C25H27N3O6S/c1-15-12-16(2)26-28(24(15)30)22(17-6-11-20-21(13-17)34-14-33-20)23(29)27-35(31,32)19-9-7-18(8-10-19)25(3,4)5/h6-13,22H,14H2,1-5H3,(H,27,29)
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n/an/a 18n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290940
PNG
(CHEMBL94929 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3,5-di...)
Show SMILES Cc1cc(C)c(=O)n(n1)C(C(=O)NS(=O)(=O)c1ccc(cc1)C(C)(C)C)c1ccc2OCOc2c1
Show InChI InChI=1S/C25H27N3O6S/c1-15-12-16(2)26-28(24(15)30)22(17-6-11-20-21(13-17)34-14-33-20)23(29)27-35(31,32)19-9-7-18(8-10-19)25(3,4)5/h6-13,22H,14H2,1-5H3,(H,27,29)
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n/an/a 20n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Compound was evaluated for the antagonism at the Endothelin A receptor (G-protein coupled endothelin A)

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290949
PNG
(CHEMBL94918 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3,5-di...)
Show SMILES CC(C)c1ccc(cc1)S(=O)(=O)NC(=O)C(c1ccc2OCOc2c1)n1nc(C)cc(C)c1=O
Show InChI InChI=1S/C24H25N3O6S/c1-14(2)17-5-8-19(9-6-17)34(30,31)26-23(28)22(27-24(29)15(3)11-16(4)25-27)18-7-10-20-21(12-18)33-13-32-20/h5-12,14,22H,13H2,1-4H3,(H,26,28)
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n/an/a 29n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Compound was evaluated for the antagonism at the Endothelin A receptor (G-protein coupled endothelin A)

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290950
PNG
(CHEMBL421563 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3-met...)
Show SMILES Cc1ccc(=O)n(n1)C(C(=O)NS(=O)(=O)c1ccc(cc1)C(C)(C)C)c1ccc2OCOc2c1
Show InChI InChI=1S/C24H25N3O6S/c1-15-5-12-21(28)27(25-15)22(16-6-11-19-20(13-16)33-14-32-19)23(29)26-34(30,31)18-9-7-17(8-10-18)24(2,3)4/h5-13,22H,14H2,1-4H3,(H,26,29)
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n/an/a 32n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290953
PNG
(CHEMBL96762 | N-[2-Benzo[1,3]dioxol-5-yl-2-(5-ethy...)
Show SMILES CCc1cc(C)nn(C(C(=O)NS(=O)(=O)c2ccc(cc2)C(C)C)c2ccc3OCOc3c2)c1=O
Show InChI InChI=1S/C25H27N3O6S/c1-5-17-12-16(4)26-28(25(17)30)23(19-8-11-21-22(13-19)34-14-33-21)24(29)27-35(31,32)20-9-6-18(7-10-20)15(2)3/h6-13,15,23H,5,14H2,1-4H3,(H,27,29)
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n/an/a 32n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290952
PNG
(CHEMBL330424 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3-met...)
Show SMILES CC(C)c1ccc(cc1)S(=O)(=O)NC(=O)C(c1ccc2OCOc2c1)n1nc(C)ccc1=O
Show InChI InChI=1S/C23H23N3O6S/c1-14(2)16-5-8-18(9-6-16)33(29,30)25-23(28)22(26-21(27)11-4-15(3)24-26)17-7-10-19-20(12-17)32-13-31-19/h4-12,14,22H,13H2,1-3H3,(H,25,28)
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n/an/a 34n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Compound was evaluated for the antagonism at the Endothelin B receptor in isolated rabbit jugularis vein

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290954
PNG
(4-[1-Benzo[1,3]dioxol-5-yl-2-(4-isopropyl-benzenes...)
Show SMILES CCCc1cc(ccc1OC(C(=O)[N-]S(=O)(=O)c1ccc(cc1)C(C)C)c1ccc2OCOc2c1)C([O-])=O
Show InChI InChI=1S/C28H29NO8S/c1-4-5-19-14-21(28(31)32)9-12-23(19)37-26(20-8-13-24-25(15-20)36-16-35-24)27(30)29-38(33,34)22-10-6-18(7-11-22)17(2)3/h6-15,17,26H,4-5,16H2,1-3H3,(H2,29,30,31,32)/p-2
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n/an/a 41n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290947
PNG
(CHEMBL328311 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3-met...)
Show SMILES COc1ccc(cc1)S(=O)(=O)NC(=O)C(c1ccc2OCOc2c1)n1nc(C)ccc1=O
Show InChI InChI=1S/C21H19N3O7S/c1-13-3-10-19(25)24(22-13)20(14-4-9-17-18(11-14)31-12-30-17)21(26)23-32(27,28)16-7-5-15(29-2)6-8-16/h3-11,20H,12H2,1-2H3,(H,23,26)
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n/an/a 160n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290955
PNG
(CHEMBL96662 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3-meth...)
Show SMILES Cc1ccc(=O)n(n1)C(C(=O)NS(=O)(=O)c1ccc(Br)cc1)c1ccc2OCOc2c1
Show InChI InChI=1S/C20H16BrN3O6S/c1-12-2-9-18(25)24(22-12)19(13-3-8-16-17(10-13)30-11-29-16)20(26)23-31(27,28)15-6-4-14(21)5-7-15/h2-10,19H,11H2,1H3,(H,23,26)
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n/an/a 230n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290939
PNG
(CHEMBL97595 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3-meth...)
Show SMILES Cc1ccc(=O)n(n1)C(C(=O)NS(=O)(=O)c1ccccc1)c1ccc2OCOc2c1
Show InChI InChI=1S/C20H17N3O6S/c1-13-7-10-18(24)23(21-13)19(14-8-9-16-17(11-14)29-12-28-16)20(25)22-30(26,27)15-5-3-2-4-6-15/h2-11,19H,12H2,1H3,(H,22,25)
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n/an/a 230n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290944
PNG
(Biphenyl-4-sulfonic acid [2-benzo[1,3]dioxol-5-yl-...)
Show SMILES Cc1ccc(=O)n(n1)C(C(=O)NS(=O)(=O)c1ccc(cc1)-c1ccccc1)c1ccc2OCOc2c1
Show InChI InChI=1S/C26H21N3O6S/c1-17-7-14-24(30)29(27-17)25(20-10-13-22-23(15-20)35-16-34-22)26(31)28-36(32,33)21-11-8-19(9-12-21)18-5-3-2-4-6-18/h2-15,25H,16H2,1H3,(H,28,31)
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n/an/a 240n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290945
PNG
(CHEMBL94654 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3-cycl...)
Show SMILES CC(C)c1ccc(cc1)S(=O)(=O)NC(=O)C(c1ccc2OCOc2c1)n1nc(ccc1=O)C1CC1
Show InChI InChI=1S/C25H25N3O6S/c1-15(2)16-5-8-19(9-6-16)35(31,32)27-25(30)24(18-7-11-21-22(13-18)34-14-33-21)28-23(29)12-10-20(26-28)17-3-4-17/h5-13,15,17,24H,3-4,14H2,1-2H3,(H,27,30)
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n/an/a 260n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290951
PNG
(CHEMBL96847 | N-[2-Benzo[1,3]dioxol-5-yl-2-(5-meth...)
Show SMILES CCCc1cc(C)c(=O)n(n1)C(C(=O)NS(=O)(=O)c1ccc(cc1)C(C)C)c1ccc2OCOc2c1
Show InChI InChI=1S/C26H29N3O6S/c1-5-6-20-13-17(4)26(31)29(27-20)24(19-9-12-22-23(14-19)35-15-34-22)25(30)28-36(32,33)21-10-7-18(8-11-21)16(2)3/h7-14,16,24H,5-6,15H2,1-4H3,(H,28,30)
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n/an/a 290n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290938
PNG
(CHEMBL94720 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3,4-di...)
Show SMILES CC(C)c1ccc(cc1)S(=O)(=O)NC(=O)C(c1ccc2OCOc2c1)n1nc(C)c(C)cc1=O
Show InChI InChI=1S/C24H25N3O6S/c1-14(2)17-5-8-19(9-6-17)34(30,31)26-24(29)23(27-22(28)11-15(3)16(4)25-27)18-7-10-20-21(12-18)33-13-32-20/h5-12,14,23H,13H2,1-4H3,(H,26,29)
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n/an/a 340n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290940
PNG
(CHEMBL94929 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3,5-di...)
Show SMILES Cc1cc(C)c(=O)n(n1)C(C(=O)NS(=O)(=O)c1ccc(cc1)C(C)(C)C)c1ccc2OCOc2c1
Show InChI InChI=1S/C25H27N3O6S/c1-15-12-16(2)26-28(24(15)30)22(17-6-11-20-21(13-17)34-14-33-20)23(29)27-35(31,32)19-9-7-18(8-10-19)25(3,4)5/h6-13,22H,14H2,1-5H3,(H,27,29)
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n/an/a 550n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Compound was evaluated for the antagonism at the Endothelin A receptor in isolated rat aortic rings

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290940
PNG
(CHEMBL94929 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3,5-di...)
Show SMILES Cc1cc(C)c(=O)n(n1)C(C(=O)NS(=O)(=O)c1ccc(cc1)C(C)(C)C)c1ccc2OCOc2c1
Show InChI InChI=1S/C25H27N3O6S/c1-15-12-16(2)26-28(24(15)30)22(17-6-11-20-21(13-17)34-14-33-20)23(29)27-35(31,32)19-9-7-18(8-10-19)25(3,4)5/h6-13,22H,14H2,1-5H3,(H,27,29)
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n/an/a 550n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290958
PNG
(CHEMBL318017 | N-[2-Benzo[1,3]dioxol-5-yl-2-(6-oxo...)
Show SMILES CCCc1ccc(=O)n(n1)C(C(=O)NS(=O)(=O)c1ccc(cc1)C(C)C)c1ccc2OCOc2c1
Show InChI InChI=1S/C25H27N3O6S/c1-4-5-19-9-13-23(29)28(26-19)24(18-8-12-21-22(14-18)34-15-33-21)25(30)27-35(31,32)20-10-6-17(7-11-20)16(2)3/h6-14,16,24H,4-5,15H2,1-3H3,(H,27,30)
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n/an/a 640n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290954
PNG
(4-[1-Benzo[1,3]dioxol-5-yl-2-(4-isopropyl-benzenes...)
Show SMILES CCCc1cc(ccc1OC(C(=O)[N-]S(=O)(=O)c1ccc(cc1)C(C)C)c1ccc2OCOc2c1)C([O-])=O
Show InChI InChI=1S/C28H29NO8S/c1-4-5-19-14-21(28(31)32)9-12-23(19)37-26(20-8-13-24-25(15-20)36-16-35-24)27(30)29-38(33,34)22-10-6-18(7-11-22)17(2)3/h6-15,17,26H,4-5,16H2,1-3H3,(H2,29,30,31,32)/p-2
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n/an/a 900n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290960
PNG
(CHEMBL96644 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3-oxo-...)
Show SMILES CC(C)c1ccc(cc1)S(=O)(=O)NC(=O)C(c1ccc2OCOc2c1)n1nc2CCCc2cc1=O
Show InChI InChI=1S/C25H25N3O6S/c1-15(2)16-6-9-19(10-7-16)35(31,32)27-25(30)24(18-8-11-21-22(12-18)34-14-33-21)28-23(29)13-17-4-3-5-20(17)26-28/h6-13,15,24H,3-5,14H2,1-2H3,(H,27,30)
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n/an/a 1.70E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290950
PNG
(CHEMBL421563 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3-met...)
Show SMILES Cc1ccc(=O)n(n1)C(C(=O)NS(=O)(=O)c1ccc(cc1)C(C)(C)C)c1ccc2OCOc2c1
Show InChI InChI=1S/C24H25N3O6S/c1-15-5-12-21(28)27(25-15)22(16-6-11-19-20(13-16)33-14-32-19)23(29)26-34(30,31)18-9-7-17(8-10-18)24(2,3)4/h5-13,22H,14H2,1-4H3,(H,26,29)
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n/an/a 2.00E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290944
PNG
(Biphenyl-4-sulfonic acid [2-benzo[1,3]dioxol-5-yl-...)
Show SMILES Cc1ccc(=O)n(n1)C(C(=O)NS(=O)(=O)c1ccc(cc1)-c1ccccc1)c1ccc2OCOc2c1
Show InChI InChI=1S/C26H21N3O6S/c1-17-7-14-24(30)29(27-17)25(20-10-13-22-23(15-20)35-16-34-22)26(31)28-36(32,33)21-11-8-19(9-12-21)18-5-3-2-4-6-18/h2-15,25H,16H2,1H3,(H,28,31)
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n/an/a 2.40E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290960
PNG
(CHEMBL96644 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3-oxo-...)
Show SMILES CC(C)c1ccc(cc1)S(=O)(=O)NC(=O)C(c1ccc2OCOc2c1)n1nc2CCCc2cc1=O
Show InChI InChI=1S/C25H25N3O6S/c1-15(2)16-6-9-19(10-7-16)35(31,32)27-25(30)24(18-8-11-21-22(12-18)34-14-33-21)28-23(29)13-17-4-3-5-20(17)26-28/h6-13,15,24H,3-5,14H2,1-2H3,(H,27,30)
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n/an/a 2.50E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290945
PNG
(CHEMBL94654 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3-cycl...)
Show SMILES CC(C)c1ccc(cc1)S(=O)(=O)NC(=O)C(c1ccc2OCOc2c1)n1nc(ccc1=O)C1CC1
Show InChI InChI=1S/C25H25N3O6S/c1-15(2)16-5-8-19(9-6-16)35(31,32)27-25(30)24(18-7-11-21-22(13-18)34-14-33-21)28-23(29)12-10-20(26-28)17-3-4-17/h5-13,15,17,24H,3-4,14H2,1-2H3,(H,27,30)
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n/an/a 2.60E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290962
PNG
(CHEMBL96234 | N-[2-Benzo[1,3]dioxol-5-yl-2-(6-oxo-...)
Show SMILES CC(C)c1ccc(cc1)S(=O)(=O)NC(=O)C(N1N=C(CCC1=O)c1ccccc1)c1ccc2OCOc2c1 |c:18|
Show InChI InChI=1S/C28H27N3O6S/c1-18(2)19-8-11-22(12-9-19)38(34,35)30-28(33)27(21-10-14-24-25(16-21)37-17-36-24)31-26(32)15-13-23(29-31)20-6-4-3-5-7-20/h3-12,14,16,18,27H,13,15,17H2,1-2H3,(H,30,33)
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n/an/a 2.60E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290953
PNG
(CHEMBL96762 | N-[2-Benzo[1,3]dioxol-5-yl-2-(5-ethy...)
Show SMILES CCc1cc(C)nn(C(C(=O)NS(=O)(=O)c2ccc(cc2)C(C)C)c2ccc3OCOc3c2)c1=O
Show InChI InChI=1S/C25H27N3O6S/c1-5-17-12-16(4)26-28(25(17)30)23(19-8-11-21-22(13-19)34-14-33-21)24(29)27-35(31,32)20-9-6-18(7-10-20)15(2)3/h6-13,15,23H,5,14H2,1-4H3,(H,27,29)
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n/an/a 2.60E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290957
PNG
(CHEMBL94426 | N-{2-Benzo[1,3]dioxol-5-yl-2-[3-(4-c...)
Show SMILES CC(C)c1ccc(cc1)S(=O)(=O)NC(=O)C(N1N=C(CCC1=O)c1ccc(Cl)cc1)c1ccc2OCOc2c1 |c:18|
Show InChI InChI=1S/C28H26ClN3O6S/c1-17(2)18-5-10-22(11-6-18)39(35,36)31-28(34)27(20-7-13-24-25(15-20)38-16-37-24)32-26(33)14-12-23(30-32)19-3-8-21(29)9-4-19/h3-11,13,15,17,27H,12,14,16H2,1-2H3,(H,31,34)
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n/an/a 2.70E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290952
PNG
(CHEMBL330424 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3-met...)
Show SMILES CC(C)c1ccc(cc1)S(=O)(=O)NC(=O)C(c1ccc2OCOc2c1)n1nc(C)ccc1=O
Show InChI InChI=1S/C23H23N3O6S/c1-14(2)16-5-8-18(9-6-16)33(29,30)25-23(28)22(26-21(27)11-4-15(3)24-26)17-7-10-19-20(12-17)32-13-31-19/h4-12,14,22H,13H2,1-3H3,(H,25,28)
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n/an/a 2.90E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290942
PNG
(CHEMBL319743 | N-{2-Benzo[1,3]dioxol-5-yl-2-[3-(4-...)
Show SMILES COc1ccc(cc1)C1=NN(C(C(=O)NS(=O)(=O)c2ccc(cc2)C(C)C)c2ccc3OCOc3c2)C(=O)CC1 |t:9|
Show InChI InChI=1S/C29H29N3O7S/c1-18(2)19-6-11-23(12-7-19)40(35,36)31-29(34)28(21-8-14-25-26(16-21)39-17-38-25)32-27(33)15-13-24(30-32)20-4-9-22(37-3)10-5-20/h4-12,14,16,18,28H,13,15,17H2,1-3H3,(H,31,34)
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n/an/a 2.90E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290946
PNG
(CHEMBL97851 | N-{2-Benzo[1,3]dioxol-5-yl-2-[3-(4-m...)
Show SMILES COc1ccc(cc1)-c1ccc(=O)n(n1)C(C(=O)NS(=O)(=O)c1ccc(cc1)C(C)C)c1ccc2OCOc2c1
Show InChI InChI=1S/C29H27N3O7S/c1-18(2)19-6-11-23(12-7-19)40(35,36)31-29(34)28(21-8-14-25-26(16-21)39-17-38-25)32-27(33)15-13-24(30-32)20-4-9-22(37-3)10-5-20/h4-16,18,28H,17H2,1-3H3,(H,31,34)
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n/an/a 3.20E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290941
PNG
(CHEMBL412865 | N-[2-Benzo[1,3]dioxol-5-yl-2-(6-oxo...)
Show SMILES CC(C)c1ccc(cc1)S(=O)(=O)NC(=O)C(N1N=C(CCC1=O)c1cccs1)c1ccc2OCOc2c1 |c:18|
Show InChI InChI=1S/C26H25N3O6S2/c1-16(2)17-5-8-19(9-6-17)37(32,33)28-26(31)25(18-7-11-21-22(14-18)35-15-34-21)29-24(30)12-10-20(27-29)23-4-3-13-36-23/h3-9,11,13-14,16,25H,10,12,15H2,1-2H3,(H,28,31)
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n/an/a 3.20E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290949
PNG
(CHEMBL94918 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3,5-di...)
Show SMILES CC(C)c1ccc(cc1)S(=O)(=O)NC(=O)C(c1ccc2OCOc2c1)n1nc(C)cc(C)c1=O
Show InChI InChI=1S/C24H25N3O6S/c1-14(2)17-5-8-19(9-6-17)34(30,31)26-23(28)22(27-24(29)15(3)11-16(4)25-27)18-7-10-20-21(12-18)33-13-32-20/h5-12,14,22H,13H2,1-4H3,(H,26,28)
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n/an/a 3.50E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290937
PNG
(CHEMBL96935 | N-{2-Benzo[1,3]dioxol-5-yl-2-[3-(4-m...)
Show SMILES COc1ccc(cc1)-c1cc(C)c(=O)n(n1)C(C(=O)NS(=O)(=O)c1ccc(cc1)C(C)C)c1ccc2OCOc2c1
Show InChI InChI=1S/C30H29N3O7S/c1-18(2)20-7-12-24(13-8-20)41(36,37)32-29(34)28(22-9-14-26-27(16-22)40-17-39-26)33-30(35)19(3)15-25(31-33)21-5-10-23(38-4)11-6-21/h5-16,18,28H,17H2,1-4H3,(H,32,34)
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n/an/a 4.00E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290956
PNG
(CHEMBL94102 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3-tert...)
Show SMILES CC(C)c1ccc(cc1)S(=O)(=O)NC(=O)C(c1ccc2OCOc2c1)n1nc(ccc1=O)C(C)(C)C
Show InChI InChI=1S/C26H29N3O6S/c1-16(2)17-6-9-19(10-7-17)36(32,33)28-25(31)24(18-8-11-20-21(14-18)35-15-34-20)29-23(30)13-12-22(27-29)26(3,4)5/h6-14,16,24H,15H2,1-5H3,(H,28,31)
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n/an/a 4.00E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290961
PNG
(CHEMBL328683 | N-{2-Benzo[1,3]dioxol-5-yl-2-[3-(3,...)
Show SMILES COc1ccc(cc1OC)C1=NN(C(C(=O)NS(=O)(=O)c2ccc(cc2)C(C)C)c2ccc3OCOc3c2)C(=O)CC1 |t:11|
Show InChI InChI=1S/C30H31N3O8S/c1-18(2)19-5-9-22(10-6-19)42(36,37)32-30(35)29(21-8-13-25-27(16-21)41-17-40-25)33-28(34)14-11-23(31-33)20-7-12-24(38-3)26(15-20)39-4/h5-10,12-13,15-16,18,29H,11,14,17H2,1-4H3,(H,32,35)
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n/an/a 4.10E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290942
PNG
(CHEMBL319743 | N-{2-Benzo[1,3]dioxol-5-yl-2-[3-(4-...)
Show SMILES COc1ccc(cc1)C1=NN(C(C(=O)NS(=O)(=O)c2ccc(cc2)C(C)C)c2ccc3OCOc3c2)C(=O)CC1 |t:9|
Show InChI InChI=1S/C29H29N3O7S/c1-18(2)19-6-11-23(12-7-19)40(35,36)31-29(34)28(21-8-14-25-26(16-21)39-17-38-25)32-27(33)15-13-24(30-32)20-4-9-22(37-3)10-5-20/h4-12,14,16,18,28H,13,15,17H2,1-3H3,(H,31,34)
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n/an/a 4.20E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290951
PNG
(CHEMBL96847 | N-[2-Benzo[1,3]dioxol-5-yl-2-(5-meth...)
Show SMILES CCCc1cc(C)c(=O)n(n1)C(C(=O)NS(=O)(=O)c1ccc(cc1)C(C)C)c1ccc2OCOc2c1
Show InChI InChI=1S/C26H29N3O6S/c1-5-6-20-13-17(4)26(31)29(27-20)24(19-9-12-22-23(14-19)35-15-34-22)25(30)28-36(32,33)21-10-7-18(8-11-21)16(2)3/h7-14,16,24H,5-6,15H2,1-4H3,(H,28,30)
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n/an/a 4.50E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290938
PNG
(CHEMBL94720 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3,4-di...)
Show SMILES CC(C)c1ccc(cc1)S(=O)(=O)NC(=O)C(c1ccc2OCOc2c1)n1nc(C)c(C)cc1=O
Show InChI InChI=1S/C24H25N3O6S/c1-14(2)17-5-8-19(9-6-17)34(30,31)26-24(29)23(27-22(28)11-15(3)16(4)25-27)18-7-10-20-21(12-18)33-13-32-20/h5-12,14,23H,13H2,1-4H3,(H,26,29)
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n/an/a 5.20E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290946
PNG
(CHEMBL97851 | N-{2-Benzo[1,3]dioxol-5-yl-2-[3-(4-m...)
Show SMILES COc1ccc(cc1)-c1ccc(=O)n(n1)C(C(=O)NS(=O)(=O)c1ccc(cc1)C(C)C)c1ccc2OCOc2c1
Show InChI InChI=1S/C29H27N3O7S/c1-18(2)19-6-11-23(12-7-19)40(35,36)31-29(34)28(21-8-14-25-26(16-21)39-17-38-25)32-27(33)15-13-24(30-32)20-4-9-22(37-3)10-5-20/h4-16,18,28H,17H2,1-3H3,(H,31,34)
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n/an/a 5.70E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290957
PNG
(CHEMBL94426 | N-{2-Benzo[1,3]dioxol-5-yl-2-[3-(4-c...)
Show SMILES CC(C)c1ccc(cc1)S(=O)(=O)NC(=O)C(N1N=C(CCC1=O)c1ccc(Cl)cc1)c1ccc2OCOc2c1 |c:18|
Show InChI InChI=1S/C28H26ClN3O6S/c1-17(2)18-5-10-22(11-6-18)39(35,36)31-28(34)27(20-7-13-24-25(15-20)38-16-37-24)32-26(33)14-12-23(30-32)19-3-8-21(29)9-4-19/h3-11,13,15,17,27H,12,14,16H2,1-2H3,(H,31,34)
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n/an/a 6.40E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290937
PNG
(CHEMBL96935 | N-{2-Benzo[1,3]dioxol-5-yl-2-[3-(4-m...)
Show SMILES COc1ccc(cc1)-c1cc(C)c(=O)n(n1)C(C(=O)NS(=O)(=O)c1ccc(cc1)C(C)C)c1ccc2OCOc2c1
Show InChI InChI=1S/C30H29N3O7S/c1-18(2)20-7-12-24(13-8-20)41(36,37)32-29(34)28(22-9-14-26-27(16-22)40-17-39-26)33-30(35)19(3)15-25(31-33)21-5-10-23(38-4)11-6-21/h5-16,18,28H,17H2,1-4H3,(H,32,34)
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n/an/a 7.70E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290958
PNG
(CHEMBL318017 | N-[2-Benzo[1,3]dioxol-5-yl-2-(6-oxo...)
Show SMILES CCCc1ccc(=O)n(n1)C(C(=O)NS(=O)(=O)c1ccc(cc1)C(C)C)c1ccc2OCOc2c1
Show InChI InChI=1S/C25H27N3O6S/c1-4-5-19-9-13-23(29)28(26-19)24(18-8-12-21-22(14-18)34-15-33-21)25(30)27-35(31,32)20-10-6-17(7-11-20)16(2)3/h6-14,16,24H,4-5,15H2,1-3H3,(H,27,30)
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n/an/a 8.40E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290948
PNG
(Benzo[1,3]dioxol-5-yl-(6-oxo-3-phenyl-5,6-dihydro-...)
Show SMILES OC(=O)C(N1N=C(CCC1=O)c1ccccc1)c1ccc2OCOc2c1 |c:5|
Show InChI InChI=1S/C19H16N2O5/c22-17-9-7-14(12-4-2-1-3-5-12)20-21(17)18(19(23)24)13-6-8-15-16(10-13)26-11-25-15/h1-6,8,10,18H,7,9,11H2,(H,23,24)
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n/an/a>1.00E+5n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290955
PNG
(CHEMBL96662 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3-meth...)
Show SMILES Cc1ccc(=O)n(n1)C(C(=O)NS(=O)(=O)c1ccc(Br)cc1)c1ccc2OCOc2c1
Show InChI InChI=1S/C20H16BrN3O6S/c1-12-2-9-18(25)24(22-12)19(13-3-8-16-17(10-13)30-11-29-16)20(26)23-31(27,28)15-6-4-14(21)5-7-15/h2-10,19H,11H2,1H3,(H,23,26)
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n/an/a>1.00E+5n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290943
PNG
(CHEMBL94732 | N-{2-Benzo[1,3]dioxol-5-yl-2-[3-(2,4...)
Show SMILES COc1ccc(C2=NN(C(C(=O)NS(=O)(=O)c3ccc(cc3)C(C)C)c3ccc4OCOc4c3)C(=O)CC2)c(OC)c1 |t:6|
Show InChI InChI=1S/C30H31N3O8S/c1-18(2)19-5-9-22(10-6-19)42(36,37)32-30(35)29(20-7-13-25-27(15-20)41-17-40-25)33-28(34)14-12-24(31-33)23-11-8-21(38-3)16-26(23)39-4/h5-11,13,15-16,18,29H,12,14,17H2,1-4H3,(H,32,35)
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n/an/a>1.00E+5n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290943
PNG
(CHEMBL94732 | N-{2-Benzo[1,3]dioxol-5-yl-2-[3-(2,4...)
Show SMILES COc1ccc(C2=NN(C(C(=O)NS(=O)(=O)c3ccc(cc3)C(C)C)c3ccc4OCOc4c3)C(=O)CC2)c(OC)c1 |t:6|
Show InChI InChI=1S/C30H31N3O8S/c1-18(2)19-5-9-22(10-6-19)42(36,37)32-30(35)29(20-7-13-25-27(15-20)41-17-40-25)33-28(34)14-12-24(31-33)23-11-8-21(38-3)16-26(23)39-4/h5-11,13,15-16,18,29H,12,14,17H2,1-4H3,(H,32,35)
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n/an/a>1.00E+5n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290941
PNG
(CHEMBL412865 | N-[2-Benzo[1,3]dioxol-5-yl-2-(6-oxo...)
Show SMILES CC(C)c1ccc(cc1)S(=O)(=O)NC(=O)C(N1N=C(CCC1=O)c1cccs1)c1ccc2OCOc2c1 |c:18|
Show InChI InChI=1S/C26H25N3O6S2/c1-16(2)17-5-8-19(9-6-17)37(32,33)28-26(31)25(18-7-11-21-22(14-18)35-15-34-21)29-24(30)12-10-20(27-29)23-4-3-13-36-23/h3-9,11,13-14,16,25H,10,12,15H2,1-2H3,(H,28,31)
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n/an/a>1.00E+5n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290956
PNG
(CHEMBL94102 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3-tert...)
Show SMILES CC(C)c1ccc(cc1)S(=O)(=O)NC(=O)C(c1ccc2OCOc2c1)n1nc(ccc1=O)C(C)(C)C
Show InChI InChI=1S/C26H29N3O6S/c1-16(2)17-6-9-19(10-7-17)36(32,33)28-25(31)24(18-8-11-20-21(14-18)35-15-34-20)29-23(30)13-12-22(27-29)26(3,4)5/h6-14,16,24H,15H2,1-5H3,(H,28,31)
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n/an/a>1.00E+5n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290959
PNG
(CHEMBL96931 | N-{2-Benzo[1,3]dioxol-5-yl-2-[3-(2,5...)
Show SMILES COc1ccc(OC)c(c1)C1=NN(C(C(=O)NS(=O)(=O)c2ccc(cc2)C(C)C)c2ccc3OCOc3c2)C(=O)CC1 |t:11|
Show InChI InChI=1S/C30H31N3O8S/c1-18(2)19-5-9-22(10-6-19)42(36,37)32-30(35)29(20-7-12-26-27(15-20)41-17-40-26)33-28(34)14-11-24(31-33)23-16-21(38-3)8-13-25(23)39-4/h5-10,12-13,15-16,18,29H,11,14,17H2,1-4H3,(H,32,35)
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n/an/a>1.00E+5n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290947
PNG
(CHEMBL328311 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3-met...)
Show SMILES COc1ccc(cc1)S(=O)(=O)NC(=O)C(c1ccc2OCOc2c1)n1nc(C)ccc1=O
Show InChI InChI=1S/C21H19N3O7S/c1-13-3-10-19(25)24(22-13)20(14-4-9-17-18(11-14)31-12-30-17)21(26)23-32(27,28)16-7-5-15(29-2)6-8-16/h3-11,20H,12H2,1-2H3,(H,23,26)
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n/an/a>1.00E+5n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290940
PNG
(CHEMBL94929 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3,5-di...)
Show SMILES Cc1cc(C)c(=O)n(n1)C(C(=O)NS(=O)(=O)c1ccc(cc1)C(C)(C)C)c1ccc2OCOc2c1
Show InChI InChI=1S/C25H27N3O6S/c1-15-12-16(2)26-28(24(15)30)22(17-6-11-20-21(13-17)34-14-33-20)23(29)27-35(31,32)19-9-7-18(8-10-19)25(3,4)5/h6-13,22H,14H2,1-5H3,(H,27,29)
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n/an/a>1.00E+5n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290939
PNG
(CHEMBL97595 | N-[2-Benzo[1,3]dioxol-5-yl-2-(3-meth...)
Show SMILES Cc1ccc(=O)n(n1)C(C(=O)NS(=O)(=O)c1ccccc1)c1ccc2OCOc2c1
Show InChI InChI=1S/C20H17N3O6S/c1-13-7-10-18(24)23(21-13)19(14-8-9-16-17(11-14)29-12-28-16)20(25)22-30(26,27)15-5-3-2-4-6-15/h2-11,19H,12H2,1H3,(H,22,25)
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n/an/a>1.00E+5n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin-1 receptor


(RAT)		BDBM50290948
PNG
(Benzo[1,3]dioxol-5-yl-(6-oxo-3-phenyl-5,6-dihydro-...)
Show SMILES OC(=O)C(N1N=C(CCC1=O)c1ccccc1)c1ccc2OCOc2c1 |c:5|
Show InChI InChI=1S/C19H16N2O5/c22-17-9-7-14(12-4-2-1-3-5-12)20-21(17)18(19(23)24)13-6-8-15-16(10-13)26-11-25-15/h1-6,8,10,18H,7,9,11H2,(H,23,24)
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n/an/a>1.00E+5n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290961
PNG
(CHEMBL328683 | N-{2-Benzo[1,3]dioxol-5-yl-2-[3-(3,...)
Show SMILES COc1ccc(cc1OC)C1=NN(C(C(=O)NS(=O)(=O)c2ccc(cc2)C(C)C)c2ccc3OCOc3c2)C(=O)CC1 |t:11|
Show InChI InChI=1S/C30H31N3O8S/c1-18(2)19-5-9-22(10-6-19)42(36,37)32-30(35)29(21-8-13-25-27(16-21)41-17-40-25)33-28(34)14-11-23(31-33)20-7-12-24(38-3)26(15-20)39-4/h5-10,12-13,15-16,18,29H,11,14,17H2,1-4H3,(H,32,35)
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n/an/a>1.00E+5n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290962
PNG
(CHEMBL96234 | N-[2-Benzo[1,3]dioxol-5-yl-2-(6-oxo-...)
Show SMILES CC(C)c1ccc(cc1)S(=O)(=O)NC(=O)C(N1N=C(CCC1=O)c1ccccc1)c1ccc2OCOc2c1 |c:18|
Show InChI InChI=1S/C28H27N3O6S/c1-18(2)19-8-11-22(12-9-19)38(34,35)30-28(33)27(21-10-14-24-25(16-21)37-17-36-24)31-26(32)15-13-23(29-31)20-6-4-3-5-7-20/h3-12,14,16,18,27H,13,15,17H2,1-2H3,(H,30,33)
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n/an/a>1.00E+5n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
Endothelin receptor type B


(Sus scrofa)		BDBM50290959
PNG
(CHEMBL96931 | N-{2-Benzo[1,3]dioxol-5-yl-2-[3-(2,5...)
Show SMILES COc1ccc(OC)c(c1)C1=NN(C(C(=O)NS(=O)(=O)c2ccc(cc2)C(C)C)c2ccc3OCOc3c2)C(=O)CC1 |t:11|
Show InChI InChI=1S/C30H31N3O8S/c1-18(2)19-5-9-22(10-6-19)42(36,37)32-30(35)29(20-7-12-26-27(15-20)41-17-40-26)33-28(34)14-11-24(31-33)23-16-21(38-3)8-13-25(23)39-4/h5-10,12-13,15-16,18,29H,11,14,17H2,1-4H3,(H,32,35)
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n/an/a>1.00E+5n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to endothelin B receptor of porcine kidney membranes

Bioorg Med Chem Lett 7: 275-280 (1997)


Article DOI: 10.1016/S0960-894X(96)00617-8
BindingDB Entry DOI: 10.7270/Q2QF8SWT
More data for this
Ligand-Target Pair
* indicates data uncertainty>20%