Found 3 hits of Enzyme Inhibition Constant Data Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Delta-type/Kappa-type/Mu-type opioid receptor
(Homo sapiens (Human)) | BDBM50223658
(CHEMBL279613)Show InChI InChI=1S/C16H23NO2/c1-4-15(18)19-16(14-8-6-5-7-9-14)10-11-17(3)13(2)12-16/h5-9,13H,4,10-12H2,1-3H3/t13-,16+/m0/s1 | PDB
UniProtKB/SwissProt
DrugBank antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet
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CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description Ability to displace [3H]etorphine from Opioid receptors in guinea pig brain |
J Med Chem 25: 9-12 (1982)
BindingDB Entry DOI: 10.7270/Q2PZ5C1C |
More data for this Ligand-Target Pair | |
Delta-type/Kappa-type/Mu-type opioid receptor
(Homo sapiens (Human)) | BDBM50223656
(CHEMBL2079647)Show InChI InChI=1S/C16H23NO2/c1-4-15(18)19-16(14-8-6-5-7-9-14)10-11-17(3)13(2)12-16/h5-9,13H,4,10-12H2,1-3H3 | PDB
UniProtKB/SwissProt
DrugBank antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description Ability to displace [3H]etorphine from Opioid receptors in guinea pig brain |
J Med Chem 25: 9-12 (1982)
BindingDB Entry DOI: 10.7270/Q2PZ5C1C |
More data for this Ligand-Target Pair | |
Delta-type/Kappa-type/Mu-type opioid receptor
(Homo sapiens (Human)) | BDBM50223657
(CHEMBL273784)Show InChI InChI=1S/C16H23NO2/c1-4-15(18)19-16(14-8-6-5-7-9-14)10-11-17(3)13(2)12-16/h5-9,13H,4,10-12H2,1-3H3/t13?,16-/m0/s1 | PDB
UniProtKB/SwissProt
DrugBank antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL PC cid PC sid UniChem
Patents
| PubMed
| n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description Ability to displace [3H]etorphine from Opioid receptors in guinea pig brain |
J Med Chem 25: 9-12 (1982)
BindingDB Entry DOI: 10.7270/Q2PZ5C1C |
More data for this Ligand-Target Pair | |