Affinity Data by PubMed id=722762

Found 2 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Sodium-dependent serotonin transporter (Rattus norvegicus (rat))	BDBM50010138 (CHEMBL3248703) Show SMILES Cl.CC(N)Cc1cc(Cl)c(Cl)s1 Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	PubMed	n/a	n/a	450	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Inhibition of SERT-mediated 5-HT uptake in Wistar rat brain synaptosomes				J Med Chem 21: 978-81 (1979) BindingDB Entry DOI: 10.7270/Q2K9392R
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium-dependent serotonin transporter (Rattus norvegicus (rat))	BDBM50029100 (2-(4-Chloro-phenyl)-1-methyl-ethylamine \| CHEMBL35...) Show SMILES CC(N)Cc1ccc(Cl)cc1 Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	500	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Inhibition of SERT-mediated 5-HT uptake in Wistar rat brain synaptosomes				J Med Chem 21: 978-81 (1979) BindingDB Entry DOI: 10.7270/Q2K9392R
TBA Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%