Affinity Data by PubMed id=8383730

PubMed code 8383730

Found 7 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Leukotriene B4 receptor 1 (Homo sapiens (Human))	BDBM50042185 (4,5-Bis-benzo[1,3]dioxol-5-ylmethyl-1-methyl-1H-im...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	1.30E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Displacement of [3H]LTB4 from LTB4 receptor expressed in human U937 cell membrane				J Nat Prod 56: 116-121 (1993) Article DOI: 10.1021/np50091a016 BindingDB Entry DOI: 10.7270/Q20K28K5
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Leukotriene B4 receptor 1 (Homo sapiens (Human))	BDBM50292405 (CHEMBL485054 \| leucettamidine) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	5.30E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Displacement of [3H]LTB4 from LTB4 receptor expressed in human U937 cell membrane				J Nat Prod 56: 116-121 (1993) Article DOI: 10.1021/np50091a016 BindingDB Entry DOI: 10.7270/Q20K28K5
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Leukotriene B4 receptor 1 (Homo sapiens (Human))	BDBM50292406 (CHEMBL485053 \| leucettamine B) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Displacement of [3H]LTB4 from LTB4 receptor expressed in human U937 cell membrane				J Nat Prod 56: 116-121 (1993) Article DOI: 10.1021/np50091a016 BindingDB Entry DOI: 10.7270/Q20K28K5
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Leukotriene B4 receptor 1 (Homo sapiens (Human))	BDBM50042185 (4,5-Bis-benzo[1,3]dioxol-5-ylmethyl-1-methyl-1H-im...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	750	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Binding affinity to LTB4 receptor in human U937 cells by whole cell assay				J Nat Prod 56: 116-121 (1993) Article DOI: 10.1021/np50091a016 BindingDB Entry DOI: 10.7270/Q20K28K5
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Leukotriene B4 receptor 1 (Homo sapiens (Human))	BDBM50042185 (4,5-Bis-benzo[1,3]dioxol-5-ylmethyl-1-methyl-1H-im...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Displacement of [3H]LTB4 from LTB4 receptor expressed in human U937 cell membrane				J Nat Prod 56: 116-121 (1993) Article DOI: 10.1021/np50091a016 BindingDB Entry DOI: 10.7270/Q20K28K5
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Leukotriene B4 receptor 1 (Homo sapiens (Human))	BDBM50042185 (4,5-Bis-benzo[1,3]dioxol-5-ylmethyl-1-methyl-1H-im...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.60E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Antagonist activity at LTB4 receptor in fura-2 loaded human U937 cells assessed as inhibition of LTB4-induced calcium mobilization				J Nat Prod 56: 116-121 (1993) Article DOI: 10.1021/np50091a016 BindingDB Entry DOI: 10.7270/Q20K28K5
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Leukotriene B4 receptor 1 (Homo sapiens (Human))	BDBM50292405 (CHEMBL485054 \| leucettamidine) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.56E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Displacement of [3H]LTB4 from LTB4 receptor expressed in human U937 cell membrane				J Nat Prod 56: 116-121 (1993) Article DOI: 10.1021/np50091a016 BindingDB Entry DOI: 10.7270/Q20K28K5
TBA Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%