Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50066481 ((S)-2-Acetylamino-N-[(5S,11R,14S,17R,19aS)-17-cycl...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description 50% reduction in myeloperoxidase secretion from human PMNs mediated by 100 nM C5a | J Med Chem 41: 3417-25 (1998) Article DOI: 10.1021/jm9800651 BindingDB Entry DOI: 10.7270/Q2C828FP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50066483 ((S)-2-Acetylamino-N-[(5S,12S,15S,18R,20aS)-18-cycl...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description 50% reduction in myeloperoxidase secretion from human PMNs mediated by 100 nM C5a | J Med Chem 41: 3417-25 (1998) Article DOI: 10.1021/jm9800651 BindingDB Entry DOI: 10.7270/Q2C828FP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50066481 ((S)-2-Acetylamino-N-[(5S,11R,14S,17R,19aS)-17-cycl...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 280 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description 50% reduction in binding of [125I]-C5a to human polymorphonuclear cells (PMNs) | J Med Chem 41: 3417-25 (1998) Article DOI: 10.1021/jm9800651 BindingDB Entry DOI: 10.7270/Q2C828FP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50066478 ((S)-1-[(S)-6-Amino-2-((S)-2-methylamino-3-phenyl-p...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description 50% reduction in myeloperoxidase secretion from human PMNs mediated by 100 nM C5a | J Med Chem 41: 3417-25 (1998) Article DOI: 10.1021/jm9800651 BindingDB Entry DOI: 10.7270/Q2C828FP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50066479 ((S)-2-[(S)-2-[(R)-2-({(S)-1-[(S)-6-Amino-2-((S)-2-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description 50% reduction in myeloperoxidase secretion from human PMNs mediated by 100 nM C5a | J Med Chem 41: 3417-25 (1998) Article DOI: 10.1021/jm9800651 BindingDB Entry DOI: 10.7270/Q2C828FP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50066482 ((S)-2-[(S)-2-[(S)-2-({(S)-1-[(S)-6-Amino-2-((S)-2-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description 50% reduction in binding of [125I]-C5a to human polymorphonuclear cells (PMNs) | J Med Chem 41: 3417-25 (1998) Article DOI: 10.1021/jm9800651 BindingDB Entry DOI: 10.7270/Q2C828FP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50066483 ((S)-2-Acetylamino-N-[(5S,12S,15S,18R,20aS)-18-cycl...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description 50% reduction in binding of [125I]-C5a to human polymorphonuclear cells (PMNs) | J Med Chem 41: 3417-25 (1998) Article DOI: 10.1021/jm9800651 BindingDB Entry DOI: 10.7270/Q2C828FP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50066479 ((S)-2-[(S)-2-[(R)-2-({(S)-1-[(S)-6-Amino-2-((S)-2-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description 50% reduction in binding of [125I]-C5a to human polymorphonuclear cells (PMNs) | J Med Chem 41: 3417-25 (1998) Article DOI: 10.1021/jm9800651 BindingDB Entry DOI: 10.7270/Q2C828FP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50066478 ((S)-1-[(S)-6-Amino-2-((S)-2-methylamino-3-phenyl-p...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description 50% reduction in binding of [125I]-C5a to human polymorphonuclear cells (PMNs) | J Med Chem 41: 3417-25 (1998) Article DOI: 10.1021/jm9800651 BindingDB Entry DOI: 10.7270/Q2C828FP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50066482 ((S)-2-[(S)-2-[(S)-2-({(S)-1-[(S)-6-Amino-2-((S)-2-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description 50% reduction in myeloperoxidase secretion from human PMNs mediated by 100 nM C5a | J Med Chem 41: 3417-25 (1998) Article DOI: 10.1021/jm9800651 BindingDB Entry DOI: 10.7270/Q2C828FP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50066480 ((S)-2-[(S)-2-[(S)-2-({(S)-1-[(S)-6-Amino-2-((S)-2-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.44E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description 50% reduction in binding of [125I]-C5a to human polymorphonuclear cells (PMNs) | J Med Chem 41: 3417-25 (1998) Article DOI: 10.1021/jm9800651 BindingDB Entry DOI: 10.7270/Q2C828FP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50012295 (CHEMBL217378 | ISHKDMQLGR | Ile-Ser-His-Lys-Asp-Me...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description 50% reduction in binding of [125I]-C5a to human polymorphonuclear cells (PMNs) | J Med Chem 41: 3417-25 (1998) Article DOI: 10.1021/jm9800651 BindingDB Entry DOI: 10.7270/Q2C828FP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C5a anaphylatoxin chemotactic receptor 1 (Homo sapiens (Human)) | BDBM50066480 ((S)-2-[(S)-2-[(S)-2-({(S)-1-[(S)-6-Amino-2-((S)-2-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description 50% reduction in myeloperoxidase secretion from human PMNs mediated by 100 nM C5a | J Med Chem 41: 3417-25 (1998) Article DOI: 10.1021/jm9800651 BindingDB Entry DOI: 10.7270/Q2C828FP | |||||||||||
More data for this Ligand-Target Pair |