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TargetInward rectifier potassium channel 13
LigandBDBM600745
Substrate/Competitorn/a
Meas. Tech.thallium-flux assay
IC50>30000±n/a nM
Citation Swale, DRFoil, LD Method for controlling hematophagous or sap-feeding arthropods US Patent US11632953 Publication Date 4/25/2023
More Info.:Get all data from this article,  Assay Method
 
Inward rectifier potassium channel 13
Name:Inward rectifier potassium channel 13
Synonyms:Inward rectifier K(+) channel Kir7.1 | KCJ13_HUMAN | KCNJ13 | Potassium channel, inwardly rectifying subfamily J member 13
Type:PROTEIN
Mol. Mass.:40527.12
Organism:Homo sapiens (Human)
Description:ChEMBL_105176
Residue:360
Sequence:
MDSSNCKVIAPLLSQRYRRMVTKDGHSTLQMDGAQRGLAYLRDAWGILMDMRWRWMMLVF
SASFVVHWLVFAVLWYVLAEMNGDLELDHDAPPENHTICVKYITSFTAAFSFSLETQLTI
GYGTMFPSGDCPSAIALLAIQMLLGLMLEAFITGAFVAKIARPKNRAFSIRFTDTAVVAH
MDGKPNLIFQVANTRPSPLTSVRVSAVLYQERENGKLYQTSVDFHLDGISSDECPFFIFP
LTYYHSITPSSPLATLLQHENPSHFELVVFLSAMQEGTGEICQRRTSYLPSEIMLHHCFA
SLLTRGSKGEYQIKMENFDKTVPEFPTPLVSKSPNRTDLDIHINGQSIDNFQISETGLTE
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  Blast E-value cutoff:
BDBM600745
n/a
NameBDBM600745
Synonyms:US11632953, Compound 1 | US11632953, Compound VU041
TypeSmall organic molecule
Emp. Form.C19H20F3N3O
Mol. Mass.363.3768
SMILESFC(F)(F)c1nn(CC(=O)N2CCCc3ccccc23)c2CCCCc12
Structure
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