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TargetAGAP001281-PB
LigandBDBM600750
Substrate/Competitorn/a
Meas. Tech.thallium-flux assay
IC50 15000±n/a nM
Citation Swale, DRFoil, LD Method for controlling hematophagous or sap-feeding arthropods US Patent US11632953 Publication Date 4/25/2023
More Info.:Get all data from this article,  Assay Method
 
AGAP001281-PB
Name:AGAP001281-PB
Synonyms:n/a
Type:Protein
Mol. Mass.:49315.66
Organism:African malaria mosquito
Description:A7UVQ1
Residue:426
Sequence:
MAAERPTLDEKKPLNRIFMRPGVIEEEPDSLDSVISNLPLTVVPSLARISTHGSAFSRQE
SVRSRALRPGTTRKYRRRAILKNGDCNIVLSKVSRQRLRFLQDIFTTLVDAQWRWTLLVF
AFSFIGSWLFFGAIWWLIAFTHGDLEEMHLPKNQEESGWKPCVFNIESYTSAFLFSIETQ
TTIGYGYRTTTEECPEAIFIMCFQSIYGVMMQAFMVGFVFAKMTRPKHRTQTLLFSKHAV
VCQRDGELSLMFRVGDMRKSHIIGANIRAQLIRTKLSREGEVMAQYQHELEVGADHCGSD
LFFIWPQIVTHRINTESPFYNMSASDLLQDRFEIVVILEGTVESTGQSTQARSSYVNTEI
LWGHRFEPIVFYNKENQVYEINYSKFNETHSVDTPLCSARELAEFYKYQDDYRNQAEDHH
HLQTPA
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  Blast E-value cutoff:
BDBM600750
n/a
NameBDBM600750
Synonyms:US11632953, Compound 8 | VU0652933
TypeSmall organic molecule
Emp. Form.C19H20F3N3O
Mol. Mass.363.3768
SMILESFC(F)(F)c1nn(CC(=O)N2CCc3ccccc3C2)c2CCCCc12
Structure
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