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TargetAGAP001281-PB
LigandBDBM600756
Substrate/Competitorn/a
Meas. Tech.thallium-flux assay
IC50 4600±n/a nM
Citation Swale, DRFoil, LD Method for controlling hematophagous or sap-feeding arthropods US Patent US11632953 Publication Date 4/25/2023
More Info.:Get all data from this article,  Assay Method
 
AGAP001281-PB
Name:AGAP001281-PB
Synonyms:n/a
Type:Protein
Mol. Mass.:49315.66
Organism:African malaria mosquito
Description:A7UVQ1
Residue:426
Sequence:
MAAERPTLDEKKPLNRIFMRPGVIEEEPDSLDSVISNLPLTVVPSLARISTHGSAFSRQE
SVRSRALRPGTTRKYRRRAILKNGDCNIVLSKVSRQRLRFLQDIFTTLVDAQWRWTLLVF
AFSFIGSWLFFGAIWWLIAFTHGDLEEMHLPKNQEESGWKPCVFNIESYTSAFLFSIETQ
TTIGYGYRTTTEECPEAIFIMCFQSIYGVMMQAFMVGFVFAKMTRPKHRTQTLLFSKHAV
VCQRDGELSLMFRVGDMRKSHIIGANIRAQLIRTKLSREGEVMAQYQHELEVGADHCGSD
LFFIWPQIVTHRINTESPFYNMSASDLLQDRFEIVVILEGTVESTGQSTQARSSYVNTEI
LWGHRFEPIVFYNKENQVYEINYSKFNETHSVDTPLCSARELAEFYKYQDDYRNQAEDHH
HLQTPA
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  Blast E-value cutoff:
BDBM600756
n/a
NameBDBM600756
Synonyms:US11632953, Compound 14 | VU0652934
TypeSmall organic molecule
Emp. Form.C18H18F3N3O2
Mol. Mass.365.3496
SMILESFC(F)(F)c1nn(CC(=O)N2CCOc3ccccc23)c2CCCCc12
Structure
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