| Reaction Details |
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 | Report a problem with these data |
| Target | Bromodomain-containing protein 9 [134-239] |
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| Ligand | BDBM310898 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | BRD9 AlphaLisa Binding Assay |
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| IC50 | 53.0±n/a nM |
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| Citation |  Albrecht, BK; Bellon, SF; Burdick, DJ; Cote, A; Crawford, T; Dakin, LA; Hsiao-Wei Tsui, V; Hewitt, MC; LeBlanc, Y; Magnuson, SR; Nasveschuk, CG; Romero, AF; Tang, Y; Taylor, AM; Wang, S Therapeutic compounds and uses thereof US Patent US10150767 Publication Date 12/11/2018 |
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| More Info.: | Get all data from this article, Assay Method |
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| Bromodomain-containing protein 9 [134-239] |
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| Name: | Bromodomain-containing protein 9 [134-239] |
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| Synonyms: | BRD9 | BRD9 (aa 134-239) | BRD9_HUMAN |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 12286.22 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q9H8M2[134-239] |
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| Residue: | 106 |
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| Sequence: | AENESTPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVAN
EYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMSK
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| BDBM310898 |
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| n/a |
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| Name | BDBM310898 |
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| Synonyms: | N,N-dimethyl-3-(6-methyl-7-oxo-1H-pyrrolo[2,3-c]pyridin-4-yl)benzamide | US10150767, Example 22 |
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| Type | Small organic molecule |
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| Emp. Form. | C17H17N3O2 |
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| Mol. Mass. | 295.3358 |
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| SMILES | CN(C)C(=O)c1cccc(c1)-c1cn(C)c(=O)c2[nH]ccc12 |
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| Structure | 
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