Reaction Details |
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Target | Interleukin-17F |
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Ligand | BDBM617614 |
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Substrate/Competitor | n/a |
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Meas. Tech. | AlphaLISA Assay |
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IC50 | 63.1±n/a nM |
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Citation | MARTIN, BP; WESTERMANN, J; KERN, OT; HOLMES, AJ; MORRISON, A; KICZUN, M; AL MASRI, M; SMITH, A; HUXLEY, A IL-17A MODULATORS US Patent US20230286943 Publication Date 9/14/2023 |
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More Info.: | Get all data from this article, Assay Method |
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Interleukin-17F |
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Name: | Interleukin-17F |
Synonyms: | Cytokine ML-1 | IL17F | IL17F_HUMAN | il-17f |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 18053.35 |
Organism: | Homo sapiens (Human) |
Description: | Q96PD4 |
Residue: | 163 |
Sequence: | MTVKTLHGPAMVKYLLLSILGLAFLSEAAARKIPKVGHTFFQKPESCPPVPGGSMKLDIG
IINENQRVSMSRNIESRSTSPWNYTVTWDPNRYPSEVVQAQCRNLGCINAQGKEDISMNS
VPIQQETLVVRRKHQGCSVSFQLEKVLVTVGCTCVTPVIHHVQ
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BDBM617614 |
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n/a |
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Name | BDBM617614 |
Synonyms: | US20230286943, Example 82 |
Type | Small organic molecule |
Emp. Form. | C25H31FN6O3 |
Mol. Mass. | 482.5504 |
SMILES | CCn1nccc1C(=O)N[C@@H](C1CCCCCC1)C(=O)Nc1ncc(cc1F)-c1c(C)noc1C |r| |
Structure |
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