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TargetInterleukin-17F
LigandBDBM617627
Substrate/Competitorn/a
Meas. Tech.AlphaLISA Assay
IC50 39.8±n/a nM
Citation MARTIN, BPWESTERMANN, JKERN, OTHOLMES, AJMORRISON, AKICZUN, MAL MASRI, MSMITH, AHUXLEY, A IL-17A MODULATORS US Patent US20230286943 Publication Date 9/14/2023
More Info.:Get all data from this article,  Assay Method
 
Interleukin-17F
Name:Interleukin-17F
Synonyms:Cytokine ML-1 | IL17F | IL17F_HUMAN | il-17f
Type:Enzyme Catalytic Domain
Mol. Mass.:18053.35
Organism:Homo sapiens (Human)
Description:Q96PD4
Residue:163
Sequence:
MTVKTLHGPAMVKYLLLSILGLAFLSEAAARKIPKVGHTFFQKPESCPPVPGGSMKLDIG
IINENQRVSMSRNIESRSTSPWNYTVTWDPNRYPSEVVQAQCRNLGCINAQGKEDISMNS
VPIQQETLVVRRKHQGCSVSFQLEKVLVTVGCTCVTPVIHHVQ
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM617627
n/a
NameBDBM617627
Synonyms:US20230286943, Example 95
TypeSmall organic molecule
Emp. Form.C24H30ClN7O2
Mol. Mass.483.994
SMILESCCn1nccc1C(=O)N[C@@H](C1CCCCCC1)C(=O)Nc1ccc(cn1)-c1c(Cl)cnn1C |r|
Structure
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