| Reaction Details |
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 | Report a problem with these data |
| Target | Monoacylglycerol lipase ABHD6 [33-337] |
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| Ligand | BDBM645023 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Evaluation of ABHD6 Enzyme Inhibitory Activity Assay |
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| IC50 | 1.000±n/a nM |
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| Citation |  YOSHIDA, A; HYAKUTAKE, R; NAGASHIMA, N; MISU, R; MORI, S ABHD6 ANTAGONIST US Patent US20240010658 Publication Date 1/11/2024 |
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| More Info.: | Get all data from this article, Assay Method |
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| Monoacylglycerol lipase ABHD6 [33-337] |
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| Name: | Monoacylglycerol lipase ABHD6 [33-337] |
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| Synonyms: | Monoacylglycerol lipase ABHD6 (33-337) |
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| Type: | Enzyme |
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| Mol. Mass.: | 34939.75 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q9BV23[33-337] |
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| Residue: | 305 |
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| Sequence: | ALIRIYYWYWRRTLGMQVRYVHHEDYQFCYSFRGRPGHKPSILMLHGFSAHKDMWLSVVK
FLPKNLHLVCVDMPGHEGTTRSSLDDLSIDGQVKRIHQFVECLKLNKKPFHLVGTSMGGQ
VAGVYAAYYPSDVSSLCLVCPAGLQYSTDNQFVQRLKELQGSAAVEKIPLIPSTPEEMSE
MLQLCSYVRFKVPQQILQGLVDVRIPHNNFYRKLFLEIVSEKSRYSLHQNMDKIKVPTQI
IWGKQDQVLDVSGADMLAKSIANCQVELLENCGHSVVMERPRKTAKLIIDFLASVHNTDN
NKKLD
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| BDBM645023 |
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| n/a |
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| Name | BDBM645023 |
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| Synonyms: | US20240010658, Example 3-10 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H21BrN6OS |
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| Mol. Mass. | 473.389 |
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| SMILES | Brc1ccc(N[C@@H]2CC[C@H]3CN(C[C@@H]23)C(=O)c2cc3nn(cc3s2)C2CC2)nn1 |r| |
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| Structure | 
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