| Reaction Details |
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 | Report a problem with these data |
| Target | Fatty acid-binding protein 5 |
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| Ligand | BDBM312405 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Time Resolved-Fluorescence Energy Transfer (TR-FRET) Assay |
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| IC50 | 20.0±n/a nM |
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| Citation |  Buettelmann, B; Ceccarelli, SM; Kuehne, H; Kuhn, B; Neidhart, W; Obst Sander, U; Richter, H Bicyclic thiophenylamide compounds US Patent US9604977 Publication Date 3/28/2017 |
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| More Info.: | Get all data from this article, Assay Method |
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| Fatty acid-binding protein 5 |
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| Name: | Fatty acid-binding protein 5 |
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| Synonyms: | FABP5 | FABP5_HUMAN | Fatty acid binding protein epidermal | Fatty acid-binding protein 5 (FABP5) |
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| Type: | Enzyme |
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| Mol. Mass.: | 15164.79 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q01469 |
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| Residue: | 135 |
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| Sequence: | MATVQQLEGRWRLVDSKGFDEYMKELGVGIALRKMGAMAKPDCIITCDGKNLTIKTESTL
KTTQFSCTLGEKFEETTADGRKTQTVCNFTDGALVQHQEWDGKESTITRKLKDGKLVVEC
VMNNVTCTRIYEKVE
|
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| BDBM312405 |
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| n/a |
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| Name | BDBM312405 |
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| Synonyms: | 2-[6,6-Difluoro-3-(4-methyl-thiazol-2-yl)-4,5,6,7-tetrahydro-benzo[b]thiophen-2-ylcarbamoyl]-cyclohex-1-enecarboxylic acid | US9604977, Example 151 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H20F2N2O3S2 |
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| Mol. Mass. | 438.511 |
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| SMILES | Cc1csc(n1)-c1c(NC(=O)C2=C(CCCC2)C(O)=O)sc2CC(F)(F)CCc12 |t:12| |
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| Structure | 
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