| Reaction Details |
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 | Report a problem with these data |
| Target | Bromodomain-containing protein 3 [51-123] |
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| Ligand | BDBM313790 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Binding Assay |
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| IC50 | <100±n/a nM |
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| Citation |  Burns, C; Garnier, J; Sharp, PP; Feutrill, J; Cuzzupe, A Benzodiazepines as bromodomain inhibitors US Patent US10167292 Publication Date 1/1/2019 |
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| More Info.: | Get all data from this article, Assay Method |
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| Bromodomain-containing protein 3 [51-123] |
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| Name: | Bromodomain-containing protein 3 [51-123] |
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| Synonyms: | BRD3 | BRD3_HUMAN | Bromodomain-containing protein 3 (BRD3)(BD1) | Bromodomain-containing protein 3 Bromo 1 domain(BRD3 BD1) | KIAA0043 | RING3L |
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| Type: | n/a |
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| Mol. Mass.: | 8887.10 |
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| Organism: | Homo sapiens (Human) |
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| Description: | BD1 (51-123 aa) of Q15059 |
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| Residue: | 73 |
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| Sequence: | WKHQFAWPFYQPVDAIKLNLPDYHKIIKNPMDMGTIKKRLENNYYWSASECMQDFNTMFT
NCYIYNKPTDDIV
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| BDBM313790 |
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| n/a |
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| Name | BDBM313790 |
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| Synonyms: | US10167292, Example 34 |
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| Type | Small organic molecule |
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| Emp. Form. | C18H17ClN4O |
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| Mol. Mass. | 340.807 |
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| SMILES | Cc1nnn2CCN(c3ccc(Cl)cc3)c3cc(CO)ccc3-c12 |
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| Structure | 
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